SCHEMBL7678586

SCHEMBL7678586

Cc1ccc(-c2ccc3c(c2)C=C(C(=O)Nc2ccc(CN4CCCCC4)cc2)CCS3)cc1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 13/20 0.52
MCHR1 Q99705 1/20 0.49
MAPT P10636 3/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
TP53 P04637 1/20 0.48
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
CCR7 P32248 1/20 0.46
CCR2 P41597 1/20 0.46
CXCR3 P49682 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5209488 0.86 CCR5 (0.69) CCR5MCHR1CCR7CCR2CXCR3
SCHEMBL7684813 0.86 CCR5 (0.53) CCR5CCR7CCR2CXCR3
SCHEMBL5208454 0.85 CCR5 (0.70) CCR5MCHR1CCR7CCR2CXCR3
SCHEMBL5206461 0.83 CCR5 (0.58) CCR5MCHR1KDM4EALDH1A1MEN1
SCHEMBL5209605 0.83 CCR5 (0.71) CCR5
Iodide SCHEMBL5209713 0.82 CCR5 (0.76) CCR5
SCHEMBL5209391 0.81 CCR5 (0.62) CCR5CCR7CCR2CXCR3
SCHEMBL5207354 0.81 CCR5 (0.70) CCR5MEN1KMT2A
SCHEMBL7678557 0.79 CCR2 (0.53) CCR5CCR7CCR2CXCR3
SCHEMBL7678558 0.79 CCR2 (0.53) CCR5CCR7CCR2CXCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6413947-B1 Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-02 US disclosed
US-6268354-B1 Pharmaceutical composition for antagonizing CCR5 comprising anilide derivative TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-07-31 US disclosed
US-6172061-B1 AIDS THERAPY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed
US-6166006-A Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-12-26 US disclosed
EP-1040103-A1 ANILIDE DERIVATIVE, PRODUCTION AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-10-04 EP disclosed
WO-1999032468-A1 ANILIDE DERIVATIVE, PRODUCTION AND USE THEREOF TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-07-01 WO disclosed