SCHEMBL7680644

SCHEMBL7680644

C[C@H](OS(=O)(=O)C(F)(F)F)C(=O)c1ccccc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.43
CES1 P23141 2/20 0.43
HPGD P15428 1/20 0.40
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
GAA P10253 2/20 0.39
KAT6A Q92794 3/20 0.39
ALDH1A1 P00352 2/20 0.39
ALOX15 P16050 1/20 0.39
POLB P06746 2/20 0.38
NPC1 O15118 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
RAB9A P51151 1/20 0.38
TP53 P04637 1/20 0.37
TSHR P16473 1/20 0.37
HTT P42858 1/20 0.37
ADRB2 P07550 1/20 0.36
ADRB1 P08588 1/20 0.36
ADRB3 P13945 1/20 0.36
PTPN1 P18031 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7680782 0.83 CES2 (0.46) CES2CES1HPGDKMT2AMEN1
SCHEMBL5702519 0.83 CXCR2 (0.39) HPGDKMT2AMEN1ALDH1A1POLB
SCHEMBL10712444 0.83 MAPT (0.42) CES2CES1HPGDKMT2AMEN1
SCHEMBL8112637 0.79 CES2 (0.43) CES2CES1HPGDKMT2AMEN1
SCHEMBL28564570 0.73 CES2 (0.47) CES2CES1HPGDKMT2AMEN1
SCHEMBL28701919 0.73 ATM (0.46) HPGDKMT2AMEN1GAAALDH1A1
SCHEMBL888679 0.71 CES2 (0.58) CES2CES1HPGDKMT2AMEN1
SCHEMBL30081009 0.71 CES2 (0.58) CES2CES1HPGDKMT2AMEN1
SCHEMBL9017503 0.71 CES2 (0.53) CES2CES1HPGDKMT2AMEN1
SCHEMBL20276639 0.71 ALDH1A1 (0.47) KMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362206-B1 FUNGICIDES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-03-26 US disclosed
EP-1033367-A2 Process for the preparation of optically active triazole derivatives and their imidazolidin-2-one intermediates TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-09-06 EP disclosed
US-6034248-A FUNGICIDES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-03-07 US disclosed
US-5677464-A Production of optically active triazole compounds and their intermediates TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-10-14 US disclosed
EP-0687672-A2 Production of optically active triazole compounds and their intermediates TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-12-20 EP disclosed