SCHEMBL7681194

SCHEMBL7681194

NC(=O)c1ccc2c(c1)Sc1ccccc1C2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
HPGD P15428 3/20 0.44
KDM4E B2RXH2 2/20 0.44
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
MAPT P10636 3/20 0.43
LMNA P02545 1/20 0.43
DRD2 P14416 1/20 0.42
ADRA1D P25100 1/20 0.42
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
HTR7 P34969 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
HTR2B P41595 1/20 0.42
HSD17B3 P37058 1/20 0.42
SRD5A2 P31213 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.40
HTT P42858 1/20 0.40
ATM Q13315 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11010368 0.90 HSD17B3 (0.48) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL27794501 0.85 SRD5A2 (0.58) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL21135535 0.84 MAPT (0.54) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL11011528 0.84 KMT2A (0.62) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL23648301 0.80 TRPA1 (0.53) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL10848340 0.80 HDAC8 (0.41) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL27791546 0.77 ALDH1A1 (0.49) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL30186307 0.76 MAPT (0.47) ALDH1A1HPGDMEN1KMT2AMAPT
SCHEMBL15846800 0.75 SRD5A2 (0.58) ALDH1A1HPGDKDM4EMEN1KMT2A
SCHEMBL9681571 0.75 SRD5A2 (0.54) ALDH1A1HPGDKDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150328329-A1 LIGANDS THAT TARGET HCV-E2 BINDING SITES ON CD81 AND THERAPEUTIC METHODS USING THEM American University of Cairo (EG) 2015-11-19 US disclosed
EP-1218336-A2 MELANIN CONCENTRATING HORMONE ANTAGONIST Takeda Chemical Industries, Ltd. (JP) 2002-07-03 EP disclosed
WO-2001021577-A2 MELANIN CONCENTRATING HORMONE ANTAGONIST TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-03-29 WO disclosed