SCHEMBL7683339

SCHEMBL7683339

Cc1c(-c2ccccc2)oc2c(C(=O)NCCCN3CCN(c4ccc(F)cc4OCC(F)(F)F)CC3)cccc2c1=O

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 11/20 0.74
ADRA1B P35368 10/20 0.74
ADRA1D P25100 9/20 0.74
HTR1A P08908 6/20 0.74
LMNA P02545 2/20 0.50
ALDH1A1 P00352 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.48
KDM4E B2RXH2 1/20 0.48
CYP1A2 P05177 1/20 0.48
CHRM2 P08172 1/20 0.48
CYP3A4 P08684 1/20 0.48
ADRA2A P08913 1/20 0.48
ADORA3 P0DMS8 1/20 0.48
CYP2D6 P10635 1/20 0.48
CHRM1 P11229 1/20 0.48
ACHE P22303 1/20 0.48
SLC6A2 P23975 1/20 0.48
PDE4A P27815 1/20 0.48
OPRM1 P35372 1/20 0.48
DRD3 P35462 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7050369 0.95 HTR1A (0.72) ADRA1AADRA1BADRA1DHTR1ALMNA
SCHEMBL7678716 0.94 HTR1A (0.81) ADRA1AADRA1BADRA1DHTR1ALMNA
SCHEMBL8876489 0.91 HTR1A (0.86) ADRA1AADRA1BADRA1DHTR1ALMNA
SCHEMBL7047929 0.90 HTR1A (0.74) ADRA1AADRA1BADRA1DHTR1ALMNA
SCHEMBL7054044 0.89 HTR1A (0.69) ADRA1AADRA1BADRA1DHTR1ALMNA
SCHEMBL7051595 0.89 ADRA1A (0.57) ADRA1AADRA1BADRA1DHTR1A
SCHEMBL8875596 0.87 HTR1A (0.86) ADRA1AADRA1BADRA1DHTR1ALMNA
SCHEMBL7689629 0.87 HTR1A (0.76) ADRA1AADRA1BADRA1DHTR1ALMNA
SCHEMBL7047569 0.87 HTR1A (0.83) ADRA1AADRA1BADRA1DHTR1ALMNA
Upidosin SCHEMBL6638869 0.85 HTR1A (1.00) ADRA1AADRA1BADRA1DHTR1ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403594-B1 UROGENTIAL INFECTIONS, ETC RECORDATI, S.A. CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 2002-06-11 US claimed