SCHEMBL7683632

SCHEMBL7683632

CCOC(O)c1nn(Cc2ccc(OC)cc2)cc1B1OC(C)(C)C(C)(C)O1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
UCHL1 P09936 1/20 0.48
AADAT Q8N5Z0 1/20 0.35
MEN1 O00255 2/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
KMT2A Q03164 2/20 0.34
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32
CACNA1G O43497 2/20 0.32
CACNA1H O95180 2/20 0.32
CACNA1I Q9P0X4 2/20 0.32
HDAC1 Q13547 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CYP19A1 P11511 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
SNCA P37840 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
ALOX15 P16050 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL370360 0.87 UCHL1 (0.47) UCHL1AADATMEN1NPC1RAB9A
SCHEMBL369012 0.83 UCHL1 (0.44) UCHL1AADATMEN1NPC1RAB9A
SCHEMBL369288 0.79 UCHL1 (0.49) UCHL1AADATMEN1NPC1RAB9A
SCHEMBL15595830 0.79 UCHL1 (0.51) UCHL1AADATMEN1NPC1RAB9A
SCHEMBL6837142 0.77 UCHL1 (0.64) UCHL1SMN1; SMN2KDM4EALDH1A1MAPT
SCHEMBL15182512 0.76 UCHL1 (0.52) UCHL1AADATMEN1NPC1RAB9A
SCHEMBL369251 0.75 UCHL1 (0.53) UCHL1AADATMEN1NPC1RAB9A
SCHEMBL20154072 0.75 UCHL1 (0.45) UCHL1AADATMEN1NPC1RAB9A
SCHEMBL1051278 0.70 UCHL1 (0.52) UCHL1MEN1NPC1RAB9AKMT2A
SCHEMBL4317065 0.69 MAPT (0.50) UCHL1MEN1NPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012006760-A1 TRICYCLIC COMPOUNDS AS ALLOSTERIC MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS MERCK SHARP & DOHME CORP. (US) 2012-01-19 WO disclosed
WO-2012008999-A2 TRICYCLIC COMPOUNDS AS ALLOSTERIC MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS MERCK SHARP & DOHME CORP. (US) 2012-01-19 WO disclosed