SCHEMBL7684232

SCHEMBL7684232

COc1ccccc1C1CCN(CCn2cnc3sc4c(c3c2=O)CNC4)CC1

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADRA1B P35368 13/20 0.54
HTR1A P08908 12/20 0.54
ADRA1D P25100 12/20 0.54
HTR1B P28222 12/20 0.54
ADRA1A P35348 12/20 0.54
P2RX3 P56373 3/20 0.49
SIRT2 Q8IXJ6 3/20 0.48
DRD2 P14416 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7670362 0.86 HTR1A (0.57) ADRA1BHTR1AADRA1DHTR1BADRA1A
SCHEMBL6994182 0.86 HTR1A (0.73) ADRA1BHTR1AADRA1DHTR1BADRA1A
SCHEMBL7675942 0.85 HTR1A (0.53) ADRA1BHTR1AADRA1DHTR1BADRA1A
Hydrochloric Acid SCHEMBL7719556 0.85 HTR1A (0.72) ADRA1BHTR1AADRA1DHTR1BADRA1A
SCHEMBL7677441 0.84 ADRA1B (0.74) ADRA1BHTR1AADRA1DHTR1BADRA1A
SCHEMBL6999823 0.84 HTR1A (0.56) ADRA1BHTR1AADRA1DHTR1BADRA1A
SCHEMBL7676939 0.82 HTR1A (0.53) ADRA1BHTR1AADRA1DHTR1BADRA1A
SCHEMBL7676264 0.78 HTR1A (0.48) ADRA1BHTR1AADRA1DHTR1BADRA1A
SCHEMBL7012836 0.78 KDM4E (0.49) ADRA1BHTR1AADRA1DHTR1BADRA1A
SCHEMBL6991454 0.77 HTR1A (0.73) ADRA1BHTR1AADRA1DHTR1BADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6387912-B1 STROKE THERAPY BASF AKTIENGESELLSCHAFT (DE) 2002-05-14 US disclosed
US-6355647-B1 INHIBIT THE SEROTONIN REUPTAKE. HYPERPROLACTINEMIA, VASOSPASMS, HYPERTENSION, GASTROINTESTINAL DISORDERS ASSOCIATED WITH MOTILITY AND SECRETION ABBOTT LABORATORIES 2002-03-12 US disclosed