SCHEMBL7684443

SCHEMBL7684443

Fc1ccc2c(c1)CCCC2N1CCCNCC1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.44
HTR2B P41595 2/20 0.44
TAAR1 Q96RJ0 1/20 0.42
CHRNA7 P36544 1/20 0.41
OPRM1 P35372 1/20 0.41
OPRD1 P41143 1/20 0.41
OPRK1 P41145 1/20 0.41
OPRL1 P41146 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7684984 0.84 CHRNA7 (0.41) TAAR1CHRNA7OPRM1OPRD1OPRK1
SCHEMBL3841615 0.81 HTR2C (0.53) HTR2CHTR2B
SCHEMBL7560367 0.81 CHRNA7 (0.65) HTR2CHTR2BTAAR1CHRNA7OPRM1
SCHEMBL6002146 0.81 HTR1A (0.45) HTR2C
SCHEMBL7526106 0.81 CHRNA7 (0.65) HTR2CHTR2BTAAR1CHRNA7OPRM1
SCHEMBL7832435 0.81 CHRNA7 (0.65) HTR2CHTR2BTAAR1CHRNA7OPRM1
SCHEMBL7563225 0.81 CHRNA7 (0.65) HTR2CHTR2BTAAR1CHRNA7OPRM1
SCHEMBL7684611 0.80 HTR1A (0.43) HTR2CCHRNA7
SCHEMBL6001682 0.77 RAD52 (0.43) HTR2C
SCHEMBL31204632 0.76 CHRNA7 (0.66) HTR2CTAAR1CHRNA7OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6417183-B1 DRUGS RELATES TO 1,4-DIAZACYCLOHEPTANES, TO PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND TO THEIR USE IN METHODS OF THERAPEUTIC TREATMENT OF NERVOUS SYSTEM DISORDERS ASTRAZENELA UK LIMITED (GB) 2002-07-09 US disclosed
EP-1060169-A1 1,4-DIAZACYCLOHEPTANE DERIVATIVES AstraZeneca AB (SE) 2000-12-20 EP disclosed
WO-1999032461-A1 1,4-DIAZACYCLOHEPTANE DERIVATIVES ASTRAZENECA UK LIMITED (GB) 1999-07-01 WO disclosed