SCHEMBL7684870

SCHEMBL7684870

CC(C)(C)OC(=O)C(N)c1ccc2c(c1)OCO2

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 4/20 0.57
HPGD P15428 2/20 0.46
KDM4E B2RXH2 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
KMT2A Q03164 4/20 0.45
CYP3A4 P08684 1/20 0.43
MEN1 O00255 3/20 0.42
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
MAPK9 P45984 1/20 0.41
ADRB2 P07550 1/20 0.41
ADRB1 P08588 1/20 0.41
ADRB3 P13945 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27537606 0.84 EDNRA (0.55) EDNRAHPGDKDM4ENPC1RAB9A
SCHEMBL14032401 0.84 EDNRA (0.54) EDNRAHPGDKDM4EKMT2ACYP3A4
SCHEMBL10204938 0.84 EDNRA (0.54) EDNRAHPGDKDM4EKMT2ACYP3A4
SCHEMBL7359562 0.83 EDNRA (0.54) EDNRAHPGDKDM4ENPC1RAB9A
SCHEMBL7502509 0.82 RAB9A (0.53) HPGDKDM4ENPC1RAB9AKMT2A
SCHEMBL27677819 0.82 PTGS1 (0.47) EDNRAKDM4ENPC1RAB9APTGS1
SCHEMBL27684645 0.82 PTGS1 (0.47) EDNRAKDM4ENPC1RAB9APTGS1
SCHEMBL2857614 0.80 EDNRA (0.48) EDNRAHPGDKDM4ENPC1RAB9A
SCHEMBL4381742 0.80 EDNRA (0.48) EDNRAHPGDKDM4ENPC1RAB9A
SCHEMBL7438336 0.80 EDNRA (0.39) EDNRAPTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6500842-B1 N-((4-CHLOROPHENYL)METHYL)-8-HYDROXY-7-QUINOLINECARBOXAMIDE ADMINISTERED AS VIRICIDES AGAINST HERPES VIRUS PHARMACIA & UPJOHN COMPANY 2002-12-31 US disclosed
US-6310211-B1 ANTI-VIRAL ACTIVITY AGAINST HERPES VIRUS, CYTOMEGALOVIRUS. MANY OF THESE COMPOUNDS ARE ALSO ACTIVE AGAINST VARICELLA ZOSTER VIRUS, EPSTEIN-BARR VIRUS, HERPES SIMPLEX VIRUS AND HUMAN HERPES VIRUS TYPE 8 PHARMACIA & UPJOHN COMPANY 2001-10-30 US disclosed
US-6252080-B1 HERPES, CYTOMEGALO VIRUS PHARMACIA & UPJOHN COMPANY 2001-06-26 US disclosed
US-6211376-B1 HERPES VIRUS, CYTOMEGALO VIRUS, VARICELLA-ZOSTER VIRUS,EPSTEIN-BARR VIRUS PHARMACIA & UPJOHN COMPANY 2001-04-03 US disclosed
EP-0927164-A1 8-HYDROXY-7-SUBSTITUTED QUINOLINES AS ANTI-VIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 1999-07-07 EP disclosed
WO-1998011073-A1 8-HYDROXY-7-SUBSTITUTED QUINOLINES AS ANTI-VIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 1998-03-19 WO disclosed