SCHEMBL7685436

SCHEMBL7685436

CN(CC=CCOc1ccc(C(=O)c2ccc(C(N)=O)cc2)cc1F)C1CC1

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LSS P48449 9/20 0.57
ACHE P22303 2/20 0.39
OPRM1 P35372 2/20 0.35
OPRK1 P41145 2/20 0.35
KCNH2 Q12809 1/20 0.35
VNN1 O95497 1/20 0.35
THRA P10827 1/20 0.34
THRB P10828 1/20 0.34
DPP4 P27487 1/20 0.34
DPP8 Q6V1X1 1/20 0.34
DPP9 Q86TI2 1/20 0.34
DPP7 Q9UHL4 1/20 0.34
OPRD1 P41143 1/20 0.34
BCHE P06276 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7685430 1.00 LSS (0.57) LSSACHEOPRM1OPRK1KCNH2
SCHEMBL7685855 0.87 LSS (0.57) LSSACHEVNN1DPP4DPP9
SCHEMBL7685852 0.87 LSS (0.57) LSSACHEVNN1DPP4DPP9
SCHEMBL7768086 0.78 VNN1 (0.40) ACHEOPRM1OPRK1KCNH2VNN1
SCHEMBL7685431 0.78 VNN1 (0.40) ACHEOPRM1OPRK1KCNH2VNN1
SCHEMBL23752312 0.73 LSS (1.00) LSS
SCHEMBL7679278 0.73 LSS (1.00) LSS
SCHEMBL3700933 0.72 LSS (0.71) LSS
SCHEMBL7684578 0.72 LSS (0.71) LSS
SCHEMBL3676963 0.69 LSS (0.52) LSSACHETHRATHRBBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441177-B1 Tertiary amines HOFFMANN-LA ROCHE INC. 2002-08-27 US claimed
EP-0778264-B1 Tertiary amines having antimycotic and cholesterol lowering activity HOFFMANN LA ROCHE (CH) 2001-07-11 EP claimed
US-6441177-B1 Tertiary amines HOFFMANN-LA ROCHE INC. 2002-08-27 US disclosed
US-6034275-A FUGICIDES; ATICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 2000-03-07 US disclosed