SCHEMBL7686232

SCHEMBL7686232

C=CCn1ccc2cccc(C(=O)OCC)c21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.46
CDC25B P30305 2/20 0.45
HSD17B10 Q99714 3/20 0.44
KDM4E B2RXH2 2/20 0.44
KMT2A Q03164 2/20 0.44
TDP1 Q9NUW8 1/20 0.43
CDC25A P30304 1/20 0.42
CDC25C P30307 1/20 0.42
ALDH1A1 P00352 2/20 0.41
HIF1A Q16665 1/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
CYP3A4 P08684 1/20 0.40
CYP1A2 P05177 1/20 0.40
LMNA P02545 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MEN1 O00255 1/20 0.39
USP2 O75604 1/20 0.39
HPGD P15428 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7679127 0.81 KMT2A (0.41) HSD17B10KMT2AALDH1A1NPC1RAB9A
SCHEMBL7689755 0.80 TSHR (0.46) TSHRCDC25BHSD17B10TDP1CDC25A
SCHEMBL7688128 0.79 TSHR (0.45) TSHRCDC25BHSD17B10TDP1CDC25A
SCHEMBL7689901 0.78 TSHR (0.44) TSHRCDC25BHSD17B10KDM4ETDP1
SCHEMBL1077377 0.75 NR4A2 (0.39) TSHRHSD17B10KDM4EKMT2AALDH1A1
SCHEMBL25010273 0.74 ADRA2A (0.46) TSHRKDM4EKMT2ANPC1RAB9A
SCHEMBL3011416 0.72 NPC1 (0.44) TSHRKMT2AALDH1A1HIF1ANPC1
SCHEMBL22800161 0.72 CYP3A4 (0.38) TSHRHSD17B10KDM4EALDH1A1NPC1
SCHEMBL7690871 0.71 PIM1 (0.41) KDM4E
SCHEMBL11270794 0.71 TSHR (0.66) TSHRCDC25BHSD17B10KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362201-B1 ANTIINFLAMMATORY AGENTS; ANTIALLERGENS MERCK & CO., INC. 2002-03-26 US disclosed
WO-2000051607-A1 3-CYCLOPROPYL AND 3-CYCLOBUTYL PYRROLIDINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 2000-09-08 WO disclosed