SCHEMBL7686835

SCHEMBL7686835

N#Cc1ccc(NC(=O)c2ccc3cccnc3c2O)c(Cl)c1

nearest known ligand 0.69

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 12/20 0.69
PKM P14618 1/20 0.60
KMT2A Q03164 2/20 0.48
MAPT P10636 1/20 0.48
PLEC Q15149 1/20 0.48
KDR P35968 3/20 0.48
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19347293 0.92 EGLN1 (0.69) EGLN1PKMKMT2AMAPTPLEC
SCHEMBL19347291 0.88 EGLN1 (0.71) EGLN1PKMKMT2AKDRALDH1A1
SCHEMBL19347365 0.87 EGLN1 (0.69) EGLN1PKMKMT2AKDRALDH1A1
SCHEMBL19347296 0.86 EGLN1 (0.71) EGLN1PKMKMT2AKDRALDH1A1
SCHEMBL7688593 0.85 EGLN1 (0.61) EGLN1KMT2AMAPTPLECKDR
SCHEMBL7691504 0.84 L3MBTL1 (0.60) EGLN1KMT2AMAPTPLECKDR
SCHEMBL19347292 0.83 EGLN1 (0.60) EGLN1PKMKMT2AKDRMEN1
SCHEMBL24460157 0.82 MEN1 (0.55) EGLN1KMT2AMAPTMEN1ALDH1A1
SCHEMBL19347366 0.82 EGLN1 (1.00) EGLN1PKMALDH1A1
SCHEMBL7684545 0.82 EGLN1 (0.68) EGLN1KMT2AMAPTPLECKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6500842-B1 N-((4-CHLOROPHENYL)METHYL)-8-HYDROXY-7-QUINOLINECARBOXAMIDE ADMINISTERED AS VIRICIDES AGAINST HERPES VIRUS PHARMACIA & UPJOHN COMPANY 2002-12-31 US claimed
EP-0927164-A1 8-HYDROXY-7-SUBSTITUTED QUINOLINES AS ANTI-VIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 1999-07-07 EP claimed
WO-1998011073-A1 8-HYDROXY-7-SUBSTITUTED QUINOLINES AS ANTI-VIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 1998-03-19 WO claimed
US-20210205292-A1 INHIBITORS OF CREB-CBP INTERACTION FOR TREATMENT OF LEUKEMIA THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2021-07-08 US disclosed
WO-2017156489-A1 INHIBITORS OF CREB-CBP INTERACTION FOR TREATMENT OF LEUKEMIA THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2017-09-14 WO disclosed
US-6500842-B1 N-((4-CHLOROPHENYL)METHYL)-8-HYDROXY-7-QUINOLINECARBOXAMIDE ADMINISTERED AS VIRICIDES AGAINST HERPES VIRUS PHARMACIA & UPJOHN COMPANY 2002-12-31 US disclosed
US-6310211-B1 ANTI-VIRAL ACTIVITY AGAINST HERPES VIRUS, CYTOMEGALOVIRUS. MANY OF THESE COMPOUNDS ARE ALSO ACTIVE AGAINST VARICELLA ZOSTER VIRUS, EPSTEIN-BARR VIRUS, HERPES SIMPLEX VIRUS AND HUMAN HERPES VIRUS TYPE 8 PHARMACIA & UPJOHN COMPANY 2001-10-30 US disclosed
US-6252080-B1 HERPES, CYTOMEGALO VIRUS PHARMACIA & UPJOHN COMPANY 2001-06-26 US disclosed
US-6211376-B1 HERPES VIRUS, CYTOMEGALO VIRUS, VARICELLA-ZOSTER VIRUS,EPSTEIN-BARR VIRUS PHARMACIA & UPJOHN COMPANY 2001-04-03 US disclosed
EP-0927164-A1 8-HYDROXY-7-SUBSTITUTED QUINOLINES AS ANTI-VIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 1999-07-07 EP disclosed
WO-1998011073-A1 8-HYDROXY-7-SUBSTITUTED QUINOLINES AS ANTI-VIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 1998-03-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210205292-A1 INHIBITORS OF CREB-CBP INTERACTION FOR TREATMENT OF LEUKEMIA CREBBP, CREB1, EP300 EGLN1 237/4885PKM 3706/4885KMT2A 916/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.