SCHEMBL7688254

SCHEMBL7688254

O=C(c1ccc(Br)cc1)c1cc(F)c(OC/C=C/CBr)cc1F

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LSS P48449 8/20 0.39
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.36
PPARD Q03181 1/20 0.36
AKR1C3 P42330 1/20 0.35
HPGD P15428 1/20 0.34
NPC1 O15118 1/20 0.34
MAPT P10636 1/20 0.34
MAPK1 P28482 1/20 0.34
HTT P42858 1/20 0.34
PTGES O14684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7688257 1.00 LSS (0.39) LSSKMT2AMEN1PTGDR2PPARD
SCHEMBL8904544 0.85 LSS (0.43) LSSKMT2AMEN1PTGDR2PPARD
SCHEMBL8047384 0.85 LSS (0.43) LSSKMT2AMEN1PTGDR2PPARD
SCHEMBL8903282 0.83 LSS (0.53) LSSKMT2AMEN1PPARDMAPT
SCHEMBL8045167 0.83 LSS (0.53) LSSKMT2AMEN1PPARDMAPT
SCHEMBL7687514 0.82 LSS (0.66) LSSKMT2AMEN1
SCHEMBL7687517 0.82 LSS (0.66) LSSKMT2AMEN1
Hydrochloric Acid SCHEMBL7684564 0.81 LSS (0.64) LSSKMT2AMEN1
SCHEMBL7767787 0.81 LSS (0.40) LSSKMT2AMEN1PPARDMAPK1
Hydrochloric Acid SCHEMBL7684573 0.81 LSS (0.64) LSSKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441177-B1 Tertiary amines HOFFMANN-LA ROCHE INC. 2002-08-27 US disclosed
EP-0778264-B1 Tertiary amines having antimycotic and cholesterol lowering activity HOFFMANN LA ROCHE (CH) 2001-07-11 EP disclosed
US-6034275-A FUGICIDES; ATICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 2000-03-07 US disclosed
US-5856503-A ANTICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 1999-01-05 US disclosed
EP-0778264-A1 Tertiary amines having antimycotic and cholesterol lowering activity F. HOFFMANN-LA ROCHE AG (CH) 1997-06-11 EP disclosed
EP-0778271-A2 Aminoalkyl-substituted benzo-heterocyclic compounds F. HOFFMANN-LA ROCHE AG (CH) 1997-06-11 EP disclosed