SCHEMBL7688501

SCHEMBL7688501

CN(C)Cc1ccc(C=Cc2ccccc2C(=O)N[C@@H](Cc2ccccc2)C(=O)CNS(=O)(=O)c2ccccc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 13/20 0.58
CTSB P07858 7/20 0.58
CTSS P25774 2/20 0.56
CTSK P43235 2/20 0.56
CTSL P07711 2/20 0.51
CASP1 P29466 1/20 0.40
KCNA5 P22460 1/20 0.40
ITGB1 P05556 1/20 0.39
ITGA4 P13612 1/20 0.39
ITGB7 P26010 1/20 0.39
MMP13 P45452 1/20 0.39
ALDH1A1 P00352 1/20 0.37
PTPN1 P18031 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7694140 0.91 CAPN1 (0.60) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7689922 0.90 CAPN1 (0.57) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7692161 0.89 CAPN1 (0.70) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7692245 0.86 CAPN1 (0.51) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7698259 0.86 CAPN1 (0.61) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7693964 0.86 CAPN1 (0.50) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7696964 0.85 CAPN1 (0.61) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7698802 0.84 CAPN1 (0.67) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7691261 0.84 CAPN1 (0.47) CAPN1CTSBCTSSCTSKCTSL
SCHEMBL7695923 0.84 ITGB1 (0.52) CAPN1CTSBCASP1KCNA5ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436925-B1 BETTER ABLE TO CROSS MEMBRANES; INHIBITORS OF CYSTEINE PROTEASES LIKE CALPAIN I AND II AND CATHEPSIN B AND L, CAN THUS BE USED TO CONTROL DISEASES ASSOCIATED WITH AN ELEVATED ACTIVITY OF CALPAIN ENZYMES OR CATHEPSIN ENZYMES ABBOTT LABORATORIES 2002-08-20 US disclosed