SCHEMBL7698802

SCHEMBL7698802

O=C(N[C@@H](Cc1ccccc1)C(=O)CNS(=O)(=O)c1ccccc1)c1ccccc1C=Cc1ccc2ccccc2c1

nearest known ligand 0.67

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 11/20 0.67
CTSB P07858 5/20 0.67
CTSL P07711 2/20 0.67
CTSS P25774 2/20 0.46
CTSK P43235 2/20 0.46
CASP1 P29466 1/20 0.41
PLAT P00750 1/20 0.39
CA2 P00918 1/20 0.39
SLC16A3 O15427 1/20 0.39
KCNA5 P22460 2/20 0.39
F2 P00734 1/20 0.39
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
KAT6A Q92794 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7690013 0.90 CAPN1 (0.68) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL7689922 0.90 CAPN1 (0.57) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL7693291 0.87 CAPN1 (0.52) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL7695839 0.86 CAPN1 (0.70) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL7693964 0.85 CAPN1 (0.50) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL7695603 0.84 CAPN1 (0.70) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL7693068 0.84 CAPN1 (0.70) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL7688501 0.84 CAPN1 (0.58) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL7691261 0.82 CAPN1 (0.47) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL7696004 0.82 CAPN1 (0.46) CAPN1CTSBCTSLCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436925-B1 BETTER ABLE TO CROSS MEMBRANES; INHIBITORS OF CYSTEINE PROTEASES LIKE CALPAIN I AND II AND CATHEPSIN B AND L, CAN THUS BE USED TO CONTROL DISEASES ASSOCIATED WITH AN ELEVATED ACTIVITY OF CALPAIN ENZYMES OR CATHEPSIN ENZYMES ABBOTT LABORATORIES 2002-08-20 US disclosed