SCHEMBL7688577

SCHEMBL7688577

COc1ccc(N2C(=O)c3ccccc3C2(C)O)cc1OC

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.46
KDM4E B2RXH2 3/20 0.46
MAPK1 P28482 2/20 0.46
NR1H3 Q13133 2/20 0.45
NR1H2 P55055 1/20 0.45
PGR P06401 1/20 0.43
ALDH1A1 P00352 2/20 0.43
GAA P10253 4/20 0.43
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
TNF P01375 2/20 0.40
RAB9A P51151 2/20 0.40
NPC1 O15118 1/20 0.40
RECQL P46063 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7696756 0.88 PDE4B (0.49)
SCHEMBL8707473 0.85 PDE4B (0.39) PARP1KDM4EMAPK1GAACYP3A4
SCHEMBL8707465 0.82 PDE4A (0.44) NR1H3NR1H2ALDH1A1CYP2C19TNF
SCHEMBL8711619 0.82 CMA1 (0.42) PARP1KDM4EMAPK1ALDH1A1GAA
SCHEMBL6589296 0.73 RXFP1 (0.66) KDM4EPGRALDH1A1CYP3A4CYP2C19
SCHEMBL8707894 0.73 PDE4B (0.45)
SCHEMBL7696865 0.73 PDE4A (0.45)
SCHEMBL7689616 0.72 NR1H3 (0.71) NR1H3NR1H2ALDH1A1
SCHEMBL17751369 0.67 ALDH1A1 (0.57) KDM4EMAPK1PGRALDH1A1CYP2C19
SCHEMBL8708638 0.67 NR1H3 (0.59) NR1H3NR1H2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002081446-A1 3-CYCLOPENTYLOXY-4-METHOXYPHENYL-ISOINDOLINONE DERIVATIVES AND THE USE THEREOF DAEWOONG CO., LTD. (KR) 2002-10-17 WO disclosed
WO-1998042666-A1 NOVEL 3,4-DIALKOXYPHENYL DERIVATIVES AND THE USE THEREOF DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 1998-10-01 WO disclosed