SCHEMBL7689397

SCHEMBL7689397

CCSC(=O)C1=C(CC)NC(c2ccccc2)=C(C(=O)O)C1CC

nearest known ligand 0.77

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 9/20 0.77
TRPV1 Q8NER1 3/20 0.60
ALDH1A1 P00352 4/20 0.37
CACNA1D Q01668 1/20 0.36
HTT P42858 1/20 0.35
GAA P10253 3/20 0.35
MEN1 O00255 1/20 0.35
PKM P14618 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7685039 0.90 ADORA3 (0.78) ADORA3TRPV1ALDH1A1CACNA1DHTT
SCHEMBL6374693 0.87 ADORA3 (1.00) ADORA3TRPV1ALDH1A1CACNA1DHTT
SCHEMBL7686684 0.86 ADORA3 (0.78) ADORA3TRPV1ALDH1A1HTTGAA
SCHEMBL8210401 0.77 ADORA3 (0.49) ADORA3TRPV1ALDH1A1CACNA1DHTT
SCHEMBL7682462 0.77 ADORA3 (0.79) ADORA3TRPV1ALDH1A1HTTGAA
SCHEMBL7689462 0.75 ADORA3 (1.00) ADORA3TRPV1ALDH1A1CACNA1DHTT
SCHEMBL7689135 0.71 ADORA3 (0.84) ADORA3TRPV1ALDH1A1GAAMEN1
SCHEMBL7682982 0.66 ADORA3 (1.00) ADORA3TRPV1ALDH1A1CACNA1DHTT
SCHEMBL7689604 0.66 ADORA3 (0.65) ADORA3TRPV1ALDH1A1CACNA1DHTT
SCHEMBL7681139 0.65 ADORA3 (1.00) ADORA3TRPV1ALDH1A1CACNA1DHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6376521-B1 ANTIINFLAMMATORY AGENTS; ANTIISCHEMIC AGENTS; CENTRAL NERVOUS SYSTEM DISORDERS THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES 2002-04-23 US disclosed
WO-2000002861-A1 A3 ADENOSINE RECEPTOR ANTAGONISTS THE UNITED STATES OF AMERICA, REPRESENTED BY SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2000-01-20 WO disclosed