SCHEMBL7690123

SCHEMBL7690123

CCOc1ccc2c(c1)CC(NC(=O)C(F)(F)F)C2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 9/20 0.43
CA2 P00918 9/20 0.43
CA12 O43570 6/20 0.43
CA7 P43166 6/20 0.43
CA14 Q9ULX7 6/20 0.43
CA9 Q16790 5/20 0.43
KDM4E B2RXH2 1/20 0.42
MTNR1A P48039 2/20 0.41
MTNR1B P49286 2/20 0.41
LMNA P02545 2/20 0.41
GAA P10253 1/20 0.41
DRD2 P14416 1/20 0.41
HTR1D P28221 1/20 0.41
DRD3 P35462 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
PAX8 Q06710 1/20 0.40
HPGD P15428 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7248144 1.00 CA1 (0.43) CA1CA2CA12CA7CA14
SCHEMBL6881171 0.81 CA1 (0.50) CA1CA2CA12CA7CA14
SCHEMBL4607263 0.80 CA1 (0.43) CA1CA2CA12CA7CA14
SCHEMBL7568637 0.78 KDM4E (0.49) KDM4EMTNR1AMTNR1BLMNAGAA
SCHEMBL7254509 0.78 LMNA (0.43) KDM4EMTNR1AMTNR1BLMNAGAA
SCHEMBL7254514 0.78 LMNA (0.43) KDM4EMTNR1AMTNR1BLMNAGAA
SCHEMBL7248408 0.78 KDM4E (0.49) KDM4EMTNR1AMTNR1BLMNAGAA
SCHEMBL4124063 0.78 CA1 (0.39) CA1CA2CA12CA7CA14
SCHEMBL29189280 0.77 CA1 (0.53) CA1CA2CA12CA7CA14
SCHEMBL4607688 0.76 MAPT (0.45) CA1CA2CA12CA7CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6462234-B2 FORMED BY REACTING O-ETHYL-L-TYROSINE WITH TRIFLUOROACETIC ANHYDRIDE, REACTING WITH LEWIS ACID, THEN QUENCHING WITH WATER PHARMACIA & UPJOHN COMPANY 2002-10-08 US claimed