SCHEMBL7690789

SCHEMBL7690789

Cc1cc(NC(=O)Nc2cccc(Cl)c2)c2ccccc2n1

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 4/20 0.67
KMT2A Q03164 7/20 0.59
MEN1 O00255 6/20 0.59
MAPT P10636 6/20 0.59
HTT P42858 4/20 0.59
NPC1 O15118 4/20 0.59
RAB9A P51151 4/20 0.59
LMNA P02545 3/20 0.59
GAA P10253 1/20 0.57
NPSR1 Q6W5P4 1/20 0.57
GRIK1 P39086 1/20 0.56
KDM4E B2RXH2 1/20 0.56
ALDH1A1 P00352 2/20 0.56
S1PR1 P21453 1/20 0.56
OPRD1 P41143 1/20 0.56
SMN1; SMN2 Q16637 2/20 0.55
OPRK1 P41145 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
GALR3 O60755 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7686561 0.90 IGF1R (0.67) IGF1RKMT2AMEN1MAPTHTT
SCHEMBL6586520 0.88 IGF1R (0.79) IGF1RKMT2AMEN1MAPTHTT
SCHEMBL6588862 0.88 IGF1R (0.77) IGF1RKMT2AMEN1MAPTHTT
SCHEMBL6592577 0.86 IGF1R (0.65) IGF1RKMT2AMEN1MAPTHTT
SCHEMBL4855474 0.85 HTT (0.75) IGF1RKMT2AMEN1MAPTHTT
SCHEMBL6590889 0.85 NPC1 (0.65) IGF1RKMT2AMEN1MAPTHTT
SCHEMBL6588400 0.84 IGF1R (0.66) IGF1RKMT2AMEN1MAPTHTT
SCHEMBL6591375 0.83 S1PR1 (0.63) IGF1RKMT2AMEN1MAPTHTT
SCHEMBL6592545 0.83 IGF1R (0.79) IGF1RKMT2AMEN1MAPTHTT
SCHEMBL6587428 0.82 IGF1R (0.70) IGF1RKMT2AMEN1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6337338-B1 INSULIN LIKE GROWTH FACTOR RECEPTOR IN MAMMALS TELIK, INC. 2002-01-08 US claimed
WO-2000035455-A1 HETEROARYL-ARYL UREAS AS IGF-1 RECEPTOR ANTAGONISTS TELIK, INC. (US) 2000-06-22 WO claimed
US-6337338-B1 INSULIN LIKE GROWTH FACTOR RECEPTOR IN MAMMALS TELIK, INC. 2002-01-08 US disclosed
WO-2000035455-A1 HETEROARYL-ARYL UREAS AS IGF-1 RECEPTOR ANTAGONISTS TELIK, INC. (US) 2000-06-22 WO disclosed