SCHEMBL7691052

SCHEMBL7691052

CC(C)(C)OC(=O)C[C@H](Nc1nnc(N)s1)C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
ALDH1A1 P00352 1/20 0.34
POLB P06746 2/20 0.33
CCNB2 O95067 1/20 0.32
CCNE2 O96020 1/20 0.32
CDK1 P06493 1/20 0.32
CDK4 P11802 1/20 0.32
CCNB1 P14635 1/20 0.32
CCND1 P24385 1/20 0.32
CCNE1 P24864 1/20 0.32
CDK2 P24941 1/20 0.32
CCNB3 Q8WWL7 1/20 0.32
CYP2D6 P10635 1/20 0.32
TDP1 Q9NUW8 3/20 0.32
MAPT P10636 2/20 0.32
GAA P10253 1/20 0.32
GLS O94925 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7691051 1.00 HTT (0.38) HTTHSD17B10CA1CA2ALDH1A1
SCHEMBL7692142 0.85 NPSR1 (0.42) ALDH1A1POLBTDP1MAPTGAA
SCHEMBL7692145 0.85 NPSR1 (0.42) ALDH1A1POLBTDP1MAPTGAA
SCHEMBL7693656 0.81 CTSS (0.38) HTTHSD17B10CA1CA2ALDH1A1
SCHEMBL7684472 0.73 TACR1 (0.50) ALDH1A1POLBTDP1MAPTGAA
SCHEMBL19365645 0.71 CYP2D6 (0.41) HTTALDH1A1POLBCYP2D6TDP1
SCHEMBL19609 0.71 CYP2D6 (0.41) HTTALDH1A1POLBCYP2D6TDP1
SCHEMBL22398849 0.69 CYP2D6 (0.42) HTTCA1CA2ALDH1A1POLB
SCHEMBL17995262 0.69 CYP2D6 (0.42) HTTCA1CA2ALDH1A1POLB
SCHEMBL7871486 0.69 CYP2D6 (0.42) HTTCA1CA2ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6500842-B1 N-((4-CHLOROPHENYL)METHYL)-8-HYDROXY-7-QUINOLINECARBOXAMIDE ADMINISTERED AS VIRICIDES AGAINST HERPES VIRUS PHARMACIA & UPJOHN COMPANY 2002-12-31 US disclosed
US-6310211-B1 ANTI-VIRAL ACTIVITY AGAINST HERPES VIRUS, CYTOMEGALOVIRUS. MANY OF THESE COMPOUNDS ARE ALSO ACTIVE AGAINST VARICELLA ZOSTER VIRUS, EPSTEIN-BARR VIRUS, HERPES SIMPLEX VIRUS AND HUMAN HERPES VIRUS TYPE 8 PHARMACIA & UPJOHN COMPANY 2001-10-30 US disclosed
US-6252080-B1 HERPES, CYTOMEGALO VIRUS PHARMACIA & UPJOHN COMPANY 2001-06-26 US disclosed
US-6211376-B1 HERPES VIRUS, CYTOMEGALO VIRUS, VARICELLA-ZOSTER VIRUS,EPSTEIN-BARR VIRUS PHARMACIA & UPJOHN COMPANY 2001-04-03 US disclosed
EP-0927164-A1 8-HYDROXY-7-SUBSTITUTED QUINOLINES AS ANTI-VIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 1999-07-07 EP disclosed
WO-1998011073-A1 8-HYDROXY-7-SUBSTITUTED QUINOLINES AS ANTI-VIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 1998-03-19 WO disclosed