SCHEMBL7691902

SCHEMBL7691902

O=C(O)CCCc1ccc2c(c1)CCC2

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRB P28702 3/20 0.56
RXRA P19793 2/20 0.56
RXRG P48443 2/20 0.56
FFAR4 Q5NUL3 8/20 0.55
CYP1A2 P05177 2/20 0.53
HDAC3 O15379 1/20 0.50
MAPK1 P28482 1/20 0.50
ADRA1A P35348 1/20 0.50
HDAC4 P56524 1/20 0.50
SLC6A3 Q01959 1/20 0.50
HDAC1 Q13547 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
HDAC7 Q8WUI4 1/20 0.50
HDAC2 Q92769 1/20 0.50
HDAC10 Q969S8 1/20 0.50
HDAC11 Q96DB2 1/20 0.50
HDAC8 Q9BY41 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
HDAC9 Q9UKV0 1/20 0.50
HDAC5 Q9UQL6 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7828378 0.98 FFAR4 (0.56) RXRBRXRARXRGFFAR4CYP1A2
SCHEMBL7698029 0.97 FFAR4 (0.55) RXRBRXRARXRGFFAR4CYP1A2
SCHEMBL27697415 0.95 RXRB (0.55) RXRBRXRARXRGFFAR4CYP1A2
SCHEMBL2728852 0.90 RXRB (0.67) RXRBRXRARXRGFFAR4ALDH1A1
SCHEMBL11111979 0.88 RXRB (0.64) RXRBRXRARXRGFFAR4ALDH1A1
SCHEMBL28813907 0.87 RXRB (0.46) RXRBRXRARXRGFFAR4SMN1; SMN2
SCHEMBL7535153 0.83 FFAR4 (0.50) RXRBRXRARXRGFFAR4CYP1A2
SCHEMBL31512087 0.83 FFAR4 (0.50) RXRBRXRARXRGFFAR4CYP1A2
SCHEMBL1115123 0.83 CYP1A2 (0.56) RXRBRXRARXRGFFAR4CYP1A2
SCHEMBL20680969 0.82 RXRA (0.57) RXRBRXRARXRGFFAR4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011096377-A1 PYRROLE COMPOUND 第一三共株式会社 (JP) 2011-08-11 WO disclosed
WO-2002024630-A1 PHARMACEUTICAL COMPOUNDS USEFUL AS MODULATORS OF ENDOCANNABINOID-MEDIATED RESPONSE ELI LILLY AND COMPANY (US) 2002-03-28 WO disclosed
EP-0769015-B1 PHOSPHONIC ACID COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-03-14 EP disclosed
US-5716944-A USEFUL AS PROPHYLACTIC AND THERAPEUTIC AGENTS OF VARIOUS METABOLIC BONE DISEASES SUCH AS OSTEOPOROSIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-10 US disclosed
EP-0769015-A1 PHOSPHONIC ACID COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1997-04-23 EP disclosed
WO-1996001267-A1 PHOSPHONIC ACID COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-01-18 WO disclosed
EP-0010347-A1 Novel substituted omega-aroyl(propionyl or butyryl)-L-prolines, pharmaceutical compositions containing them and processes for their preparation AMERICAN CYANAMID COMPANY (US) 1980-04-30 EP disclosed