SCHEMBL7693291

SCHEMBL7693291

CCCCC(NC(=O)c1ccccc1C=Cc1ccc2ccccc2c1)C(=O)CNS(=O)(=O)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 10/20 0.52
CTSB P07858 6/20 0.52
CTSL P07711 2/20 0.52
CTSS P25774 2/20 0.39
CTSK P43235 2/20 0.39
PYGL P06737 1/20 0.38
CYP2C9 P11712 1/20 0.38
SLC16A3 O15427 3/20 0.37
CCKBR P32239 1/20 0.37
KAT6A Q92794 1/20 0.37
MMP1 P03956 1/20 0.36
MMP7 P09237 1/20 0.36
ACE P12821 1/20 0.36
MMP12 P39900 1/20 0.36
MMP13 P45452 1/20 0.36
CASP1 P29466 1/20 0.36
TACR3 P29371 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7695233 0.90 CAPN1 (0.54) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL7690746 0.88 CAPN1 (0.56) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL7698802 0.87 CAPN1 (0.67) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL7695407 0.86 CTSB (0.50) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL7697322 0.85 CAPN1 (0.54) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL7696690 0.85 CAPN1 (0.54) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL7692161 0.85 CAPN1 (0.70) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL7697236 0.83 CAPN1 (0.51) CAPN1CTSBCTSLCTSSCTSK
SCHEMBL7695268 0.83 CTSB (0.44) CAPN1CTSBCTSSCTSKCASP1
SCHEMBL7690197 0.82 CAPN1 (0.51) CAPN1CTSBCTSLCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436925-B1 BETTER ABLE TO CROSS MEMBRANES; INHIBITORS OF CYSTEINE PROTEASES LIKE CALPAIN I AND II AND CATHEPSIN B AND L, CAN THUS BE USED TO CONTROL DISEASES ASSOCIATED WITH AN ELEVATED ACTIVITY OF CALPAIN ENZYMES OR CATHEPSIN ENZYMES ABBOTT LABORATORIES 2002-08-20 US disclosed