SCHEMBL7696947

SCHEMBL7696947

CCN1CCCC1CN(C(N)=O)c1ccc(-c2n[nH]c3c2Cc2ccccc2-3)cc1

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KDR P35968 7/20 0.47
CHEK1 O14757 11/20 0.46
CDK1 P06493 1/20 0.42
CDK2 P24941 1/20 0.42
OPRD1 P41143 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7836430 0.80 CHEK1 (0.49) KDRCHEK1CDK1CDK2
SCHEMBL7698793 0.79 RAB9A (0.48) KDRCHEK1CDK1CDK2OPRD1
SCHEMBL7094187 0.78 CHEK1 (0.53) KDRCHEK1CDK1CDK2
SCHEMBL7835370 0.78 CHEK1 (0.51) KDRCHEK1CDK1CDK2
SCHEMBL7840336 0.78 CHEK1 (0.57) KDRCHEK1CDK1CDK2
SCHEMBL7094279 0.77 KDR (0.58) KDRCHEK1CDK1CDK2
SCHEMBL7184665 0.77 CHEK1 (0.51) KDRCHEK1CDK1CDK2
SCHEMBL7832418 0.77 CHEK1 (0.51) KDRCHEK1CDK1CDK2
SCHEMBL7832382 0.76 CHEK1 (0.52) KDRCHEK1CDK1CDK2
SCHEMBL7832987 0.75 CHEK1 (0.54) KDRCHEK1CDK1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6462036-B1 INHIBITING SIGNAL TRANSDUCTION BY MODULATING ACTIVITY OF RECEPTOR AND NONRECEPTOR TYROSINE AND SERINE/THREONINE KINASES TO REGULATE AND MODULATE ABNORMAL OR INAPPROPRIATE CELL PROLIFERATION, DIFFERENTIATION, OR METABOLISM BASF AKTIENGESELLSCHAFT (DE) 2002-10-08 US disclosed