SCHEMBL7697277

SCHEMBL7697277

CCCC[C@H](NC(=O)c1ccccc1C=Cc1ccccn1)C(=O)CNC(C)=O

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 9/20 0.47
CTSB P07858 5/20 0.47
CTSK P43235 4/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36
CTSS P25774 2/20 0.35
CTSL P07711 1/20 0.35
PREP P48147 1/20 0.35
FAP Q12884 1/20 0.35
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HSPA5 P11021 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7693965 0.91 CAPN1 (0.46) CAPN1CTSBCTSKCYP1A2CYP2C19
SCHEMBL7696167 0.86 CAPN1 (0.57) CAPN1CTSBCTSKCTSSCTSL
SCHEMBL7696533 0.85 CAPN1 (0.48) CAPN1CTSBCTSKCTSSCTSL
SCHEMBL7695268 0.84 CTSB (0.44) CAPN1CTSBCTSKCTSS
SCHEMBL7696690 0.81 CAPN1 (0.54) CAPN1CTSBCTSKCTSSCTSL
SCHEMBL7376391 0.80 CAPN1 (0.49) CAPN1CTSBCTSKCTSL
SCHEMBL7689896 0.80 CAPN1 (0.75) CAPN1CTSBCTSKCTSSCTSL
SCHEMBL7696610 0.79 CAPN1 (0.58) CAPN1CTSBCTSKCYP1A2CTSS
SCHEMBL7690894 0.79 CAPN1 (0.58) CAPN1CTSBCTSKCYP1A2CTSS
Hydrochloric Acid SCHEMBL7789980 0.79 CAPN1 (0.48) CAPN1CTSBCTSKCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436925-B1 BETTER ABLE TO CROSS MEMBRANES; INHIBITORS OF CYSTEINE PROTEASES LIKE CALPAIN I AND II AND CATHEPSIN B AND L, CAN THUS BE USED TO CONTROL DISEASES ASSOCIATED WITH AN ELEVATED ACTIVITY OF CALPAIN ENZYMES OR CATHEPSIN ENZYMES ABBOTT LABORATORIES 2002-08-20 US disclosed