SCHEMBL7697291

SCHEMBL7697291

COC(=O)CN1CCC(Nc2cc(Nc3cc(Cl)c(N)c(Cl)c3)ncn2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 2/20 0.39
NOS1 P29475 5/20 0.38
NOS2 P35228 5/20 0.38
EGFR P00533 5/20 0.38
ABL1 P00519 4/20 0.38
SRC P12931 4/20 0.38
ABL2 P42684 4/20 0.38
LCK P06239 1/20 0.38
PRCP P42785 1/20 0.38
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
NOS3 P29474 3/20 0.36
FGFR1 P11362 1/20 0.36
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
FGFR3 P22607 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTR4 Q13639 1/20 0.35
MAP4K4 O95819 1/20 0.35
WNT1 P04628 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7696303 0.88 ABL1 (0.38) NOS1NOS2EGFRABL1SRC
SCHEMBL7691002 0.86 ERBB2 (0.48) EGFRMEN1KMT2AERBB2
SCHEMBL7851398 0.83 EGFR (0.50) NOS1NOS2EGFRABL1PRCP
SCHEMBL7850948 0.81 EGFR (0.47) NOS1NOS2EGFRABL1MEN1
SCHEMBL7689040 0.80 EGFR (0.47) NOS1NOS2EGFRNOS3
SCHEMBL7696986 0.80 EGFR (0.51) EGFRABL1SRCABL2LCK
SCHEMBL7844069 0.79 EGFR (0.45) NOS1NOS2EGFRABL1SRC
SCHEMBL7575605 0.79 EGFR (0.55) EGFRERBB2
SCHEMBL7851215 0.77 EGFR (0.44) NOS1NOS2EGFRNOS3
SCHEMBL7843657 0.77 EGFR (0.48) EGFRABL1SRCLCKWNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2002539214-A 2002-11-19 JP claimed
EP-1163242-A2 BICYCLIC HETEROCYCLES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESSES FOR PREPARING THEM Boehringer Ingelheim Pharma KG (DE) 2001-12-19 EP claimed
WO-2000055162-A2 BICYCLIC HETEROCYCLES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESSES FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-09-21 WO claimed