SCHEMBL7691002

SCHEMBL7691002

COC(=O)CN1CCC(Nc2cc(Nc3ccc(F)c(Cl)c3)ncn2)CC1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 3/20 0.48
EGFR P00533 14/20 0.47
KCNH2 Q12809 1/20 0.45
HPGD P15428 2/20 0.44
HTT P42858 1/20 0.44
ERBB4 Q15303 1/20 0.43
MEN1 O00255 1/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7853572 0.91 ERBB2 (0.44) ERBB2EGFRKCNH2HPGDHTT
SCHEMBL7853506 0.91 EGFR (0.46) ERBB2EGFRKCNH2HPGDHTT
SCHEMBL7855912 0.90 ERBB2 (0.45) ERBB2EGFRKCNH2HPGDHTT
SCHEMBL7853909 0.89 EGFR (0.45) ERBB2EGFRKCNH2HPGDHTT
SCHEMBL7852464 0.89 NOS1 (0.47) ERBB2EGFRKCNH2HPGDHTT
SCHEMBL7854005 0.89 HPGD (0.46) ERBB2EGFRKCNH2HPGDHTT
SCHEMBL7851398 0.87 EGFR (0.50) ERBB2EGFRHTTMEN1MAPT
SCHEMBL7697291 0.86 S1PR1 (0.39) ERBB2EGFRMEN1KMT2A
SCHEMBL7584450 0.86 ERBB2 (0.59) ERBB2EGFRERBB4MEN1KMT2A
SCHEMBL7852723 0.84 EGFR (0.47) ERBB2EGFRKCNH2HPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2002539214-A 2002-11-19 JP claimed
EP-1163242-A2 BICYCLIC HETEROCYCLES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESSES FOR PREPARING THEM Boehringer Ingelheim Pharma KG (DE) 2001-12-19 EP claimed
WO-2000055162-A2 BICYCLIC HETEROCYCLES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESSES FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-09-21 WO claimed
EP-1163242-A2 BICYCLIC HETEROCYCLES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESSES FOR PREPARING THEM Boehringer Ingelheim Pharma KG (DE) 2001-12-19 EP disclosed
WO-2000055162-A2 BICYCLIC HETEROCYCLES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESSES FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-09-21 WO disclosed