SCHEMBL7698264

SCHEMBL7698264

O=C(O)NC1CNCCc2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.51
HTR2C P28335 1/20 0.51
HTR2B P41595 1/20 0.51
TAAR1 Q96RJ0 1/20 0.51
TSHR P16473 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
HTT P42858 1/20 0.47
TAS1R3 Q7RTX0 2/20 0.46
TAS1R1 Q7RTX1 2/20 0.46
TAS1R2 Q8TE23 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
OPRM1 P35372 1/20 0.43
DRD2 P14416 2/20 0.43
DRD1 P21728 2/20 0.43
ALDH1A1 P00352 1/20 0.43
EPHX1 P07099 1/20 0.42
PRCP P42785 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL191727 0.79 HTT (0.60) HTTTAS1R3TAS1R1TAS1R2SMN1; SMN2
SCHEMBL3421659 0.79 HTT (0.60) HTTTAS1R3TAS1R1TAS1R2SMN1; SMN2
SCHEMBL191726 0.79 HTT (0.60) HTTTAS1R3TAS1R1TAS1R2SMN1; SMN2
SCHEMBL9011724 0.76 HTT (0.75) TSHRHTTTAS1R3TAS1R1TAS1R2
SCHEMBL4751069 0.76 HTR2C (0.56) HTR2AHTR2CHTR2BTAAR1TSHR
SCHEMBL23091569 0.75 TSHR (0.58) TSHRNPSR1HTTSMN1; SMN2MEN1
SCHEMBL8319836 0.75 TSHR (0.58) TSHRNPSR1HTTSMN1; SMN2MEN1
Malonic Acid SCHEMBL174816 0.74 HTR2C (0.74) HTR2AHTR2CHTR2BTAAR1TSHR
SCHEMBL25037806 0.73 SETD2 (0.49) TAS1R3TAS1R1TAS1R2DRD2
SCHEMBL21739663 0.72 TAS1R3 (0.37) HTR2AHTR2CHTR2BTAAR1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002057258-A1 CYCLO`D!AZEPANE DERIVATIVES WHICH ARE USED AS FARNESYLTRANSFERASE INHIBITORS AND METHOD FOR THE PREPARATION THEREOF LES LABORATOIRES SERVIER (FR) 2002-07-25 WO disclosed