SCHEMBL7698381

SCHEMBL7698381

COC(=O)c1ccc2c(c1)CC[C@H](CN(C)CC(=O)OCc1ccccc1)[C@@H]2c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 1/20 0.59
ALDH1A1 P00352 5/20 0.40
MAPT P10636 3/20 0.40
RAB9A P51151 3/20 0.40
KDM4E B2RXH2 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
MTNR1A P48039 2/20 0.39
MTNR1B P49286 2/20 0.39
LMNA P02545 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
ACHE P22303 1/20 0.36
HPGD P15428 3/20 0.36
CYP3A4 P08684 1/20 0.36
TACR1 P25103 1/20 0.36
TSHR P16473 2/20 0.36
NPC1 O15118 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7706981 1.00 SLC6A9 (0.59) SLC6A9ALDH1A1MAPTRAB9AKDM4E
Hydrochloric Acid SCHEMBL7708945 0.88 SLC6A9 (0.73) SLC6A9ALDH1A1MAPTKDM4EMTNR1A
Hydrochloric Acid SCHEMBL7698457 0.86 SLC6A9 (0.77) SLC6A9MTNR1AMTNR1B
SCHEMBL7700190 0.80 SLC6A9 (0.65) SLC6A9MAPTMAPK1
SCHEMBL7700569 0.78 SLC6A9 (0.81) SLC6A9MTNR1AMTNR1BMEN1KMT2A
SCHEMBL7409984 0.78 MTNR1A (0.52) SLC6A9MAPTRAB9AMTNR1AMTNR1B
Hydrochloric Acid SCHEMBL7706317 0.77 MTNR1A (0.51) SLC6A9MAPTRAB9AMTNR1AMTNR1B
Hydrochloric Acid SCHEMBL7706314 0.77 MTNR1A (0.51) SLC6A9MAPTRAB9AMTNR1AMTNR1B
Hydrochloric Acid SCHEMBL7706319 0.77 MTNR1A (0.51) SLC6A9MAPTRAB9AMTNR1AMTNR1B
SCHEMBL7700589 0.77 SLC6A9 (0.62) SLC6A9ALDH1A1MAPTKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100769-B1 AMINOMETHYLCARBOXYLIC ACID DERIVATIVES AKZO NOBEL NV (NL) 2002-12-04 EP disclosed
US-6410592-B1 THERAPY FOR CENTRAL NERVOUS SYSTEM DISORDERS, PSYCHOLOGICAL DISORDERS AKZO NOBEL N.V. (NL) 2002-06-25 US disclosed