SCHEMBL7698653

SCHEMBL7698653

Clc1cc(-c2ccccc2)ccc1CCBr

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.50
ERCC5 P28715 1/20 0.41
FEN1 P39748 1/20 0.41
CYP1A2 P05177 1/20 0.41
MME P08473 4/20 0.41
ACE P12821 3/20 0.41
PTPN1 P18031 1/20 0.40
GSK3B P49841 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
AHR P35869 1/20 0.38
HIF1A Q16665 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPK1 P28482 1/20 0.37
ALOX5 P09917 1/20 0.36
S1PR1 P21453 1/20 0.36
NR1H2 P55055 1/20 0.36
MAOB P27338 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5215840 0.86 ESR2 (0.52) ESR2ERCC5FEN1CYP1A2MME
SCHEMBL456713 0.81 ESR2 (0.50) ESR2ERCC5FEN1CYP1A2MME
SCHEMBL6308178 0.80 ESR2 (0.53) ESR2ERCC5FEN1CYP1A2MME
SCHEMBL8167859 0.79 ALDH1A1 (0.40) PTPN1GSK3BTDP1ALDH1A1MAPK1
SCHEMBL28025195 0.79 DAO (0.46) PTPN1GSK3BMAOB
SCHEMBL458111 0.78 ESR2 (0.52) ESR2ERCC5FEN1CYP1A2MME
SCHEMBL6299131 0.78 ESR2 (0.57) ESR2ERCC5FEN1CYP1A2MME
Benzene SCHEMBL28092155 0.77 TAAR1 (0.58) TDP1HIF1A
SCHEMBL8024134 0.77 MME (0.50) ESR2ERCC5FEN1MMEACE
SCHEMBL28940878 0.77 ESR2 (0.46) ESR2CYP1A2MMEACEHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216996-A2 Method to synthesise biphenylyl derivatives SANOFI-SYNTHELABO (FR) 2002-06-26 EP disclosed
CN-1335847-A Sulfonamide compound and pharmaceutical use thereof FUJISAWA PHARMACEUTICAL CO (JP) 2002-02-13 CN disclosed
CN-1268942-A Sulfonamide compounds and medicinal use thereof FUJISAWA PHARMACEUTICAL CO (JP) 2000-10-04 CN disclosed
EP-0837848-A1 4-ARYL-1-PHENYLALKYL-1,2,3,6-TETRAHYDROPYRIDINES HAVING NEUROTROPHIC AND NEUROPROTECTIVE ACTIVITY SANOFI (FR) 1998-04-29 EP disclosed
WO-1997001536-A1 4-ARYL-1-PHENYLALKYL-1,2,3,6-TETRAHYDROPYRIDINES HAVING NEUROTROPHIC AND NEUROPROTECTIVE ACTIVITY SANOFI (FR) 1997-01-16 WO disclosed