SCHEMBL7699065

SCHEMBL7699065

CC(C)(C)OC(=O)NC(=O)[C@@H](Cc1ccccc1)NC1CCN(Cc2ccccc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACE P12821 1/20 0.48
KMT2A Q03164 4/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
MEN1 O00255 1/20 0.47
DRD4 P21917 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
MAPK1 P28482 1/20 0.47
SIGMAR1 Q99720 1/20 0.46
CTSS P25774 2/20 0.46
CTSL P07711 1/20 0.46
CTSB P07858 1/20 0.46
CTSK P43235 1/20 0.46
DPP7 Q9UHL4 1/20 0.46
TP53 P04637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3957212 1.00 ACE (0.48) ACEKMT2ACYP3A4CYP2D6CYP2C9
SCHEMBL3957208 0.84 SCN9A (0.58) ACEKMT2AMEN1SIGMAR1CTSS
SCHEMBL915402 0.80 KMT2A (0.65) KMT2AMEN1DRD4L3MBTL1SIGMAR1
SCHEMBL3635817 0.79 KMT2A (0.56) KMT2AMEN1DRD4L3MBTL1SIGMAR1
SCHEMBL3960093 0.78 SIGMAR1 (0.56) KMT2ACYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL2311994 0.77 MEN1 (0.52) KMT2ACYP2D6CYP2C9CYP2C19MEN1
SCHEMBL15809950 0.77 KMT2A (0.62) ACEKMT2ACYP3A4CYP2D6CYP2C9
SCHEMBL7549641 0.77 KCNA3 (0.59) KMT2AMEN1DRD4L3MBTL1SIGMAR1
SCHEMBL1361202 0.77 KMT2A (0.62) ACEKMT2ACYP3A4CYP2D6CYP2C9
SCHEMBL3593211 0.76 KDM4E (0.58) KMT2AMEN1DRD4L3MBTL1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344449-B1 HEADACHE AND MORPHINE DEPENDENCE DR. KARL THOMAE GMBH (DE) 2002-02-05 US disclosed