SCHEMBL7699151

SCHEMBL7699151

Cn1ncc(CN2CCOCC2)c1C1NCCc2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.41
CYP2A13 Q16696 4/20 0.40
PRCP P42785 6/20 0.39
RECQL P46063 1/20 0.38
GAA P10253 1/20 0.38
DRD4 P21917 2/20 0.37
DRD3 P35462 1/20 0.37
GID4 Q8IVV7 1/20 0.36
TMEM97 Q5BJF2 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
HTR1A P08908 1/20 0.35
DRD2 P14416 1/20 0.35
HTR1D P28221 1/20 0.35
HTR2A P28223 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7699153 1.00 OPRM1 (0.41) OPRM1CYP2A13PRCPRECQLGAA
SCHEMBL8509848 0.82 CYP2A13 (0.40) CYP2A13GAADRD4DRD3TMEM97
SCHEMBL7702406 0.79 OPRM1 (0.41) OPRM1CYP2A13PRCPRECQLGAA
SCHEMBL7702411 0.79 OPRM1 (0.41) OPRM1CYP2A13PRCPRECQLGAA
SCHEMBL7702359 0.77 OPRM1 (0.41) OPRM1CYP2A13PRCPRECQLGAA
SCHEMBL7704232 0.77 PRCP (0.41) OPRM1CYP2A13PRCPRECQLGAA
SCHEMBL7704233 0.77 PRCP (0.41) OPRM1CYP2A13PRCPRECQLGAA
SCHEMBL7702361 0.77 OPRM1 (0.41) OPRM1CYP2A13PRCPRECQLGAA
SCHEMBL7697817 0.75 CYP2A13 (0.34) CYP2A13PRCPGAADRD4DRD3
SCHEMBL7703162 0.74 PRCP (0.57) OPRM1PRCPRECQLGAAGID4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901488-B1 2,4-DIAMINOPYRIMIDINE DERIVATIVES BASILEA PHARMACEUTICA AG (CH) 2002-11-06 EP disclosed
EP-0901488-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-03-17 EP disclosed
US-5866583-A Substituted 2,4-diaminopyrimidines HOFFMANN-LA ROCHE INC. (US) 1999-02-02 US disclosed
WO-1997043277-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-11-20 WO disclosed