SCHEMBL7702406

SCHEMBL7702406

Cn1cc(CN2CCOCC2)c(C2NCCc3ccccc32)n1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.41
CYP2A13 Q16696 4/20 0.40
ALDH1A1 P00352 2/20 0.39
PRCP P42785 6/20 0.39
RECQL P46063 1/20 0.38
GAA P10253 1/20 0.38
LMNA P02545 1/20 0.37
POLB P06746 1/20 0.37
KMT2A Q03164 1/20 0.37
GID4 Q8IVV7 1/20 0.36
NPC1 O15118 1/20 0.35
TP53 P04637 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7702411 1.00 OPRM1 (0.41) OPRM1CYP2A13ALDH1A1PRCPRECQL
SCHEMBL8510483 0.82 CYP2A13 (0.40) CYP2A13ALDH1A1GAALMNAPOLB
SCHEMBL7699151 0.79 OPRM1 (0.41) OPRM1CYP2A13PRCPRECQLGAA
SCHEMBL7699153 0.79 OPRM1 (0.41) OPRM1CYP2A13PRCPRECQLGAA
SCHEMBL7704233 0.77 PRCP (0.41) OPRM1CYP2A13PRCPRECQLGAA
SCHEMBL7702361 0.77 OPRM1 (0.41) OPRM1CYP2A13ALDH1A1PRCPRECQL
SCHEMBL7704232 0.77 PRCP (0.41) OPRM1CYP2A13PRCPRECQLGAA
SCHEMBL7702359 0.77 OPRM1 (0.41) OPRM1CYP2A13ALDH1A1PRCPRECQL
SCHEMBL7705571 0.75 ALDH1A1 (0.35) CYP2A13ALDH1A1PRCPGAALMNA
SCHEMBL7703162 0.74 PRCP (0.57) OPRM1PRCPRECQLGAAGID4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901488-B1 2,4-DIAMINOPYRIMIDINE DERIVATIVES BASILEA PHARMACEUTICA AG (CH) 2002-11-06 EP disclosed
EP-0901488-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-03-17 EP disclosed
US-5866583-A Substituted 2,4-diaminopyrimidines HOFFMANN-LA ROCHE INC. (US) 1999-02-02 US disclosed
WO-1997043277-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-11-20 WO disclosed