SCHEMBL7699618

SCHEMBL7699618

COCC1(C)CCOc2ccc(C=Cc3ccccc3C(=O)O)cc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 1/20 0.42
GRIA1 P42261 1/20 0.42
GRIA2 P42262 1/20 0.42
GRIA3 P42263 1/20 0.42
GRIA4 P48058 1/20 0.42
GRIK2 Q13002 1/20 0.42
GRIK3 Q13003 1/20 0.42
RARA P10276 5/20 0.40
RARB P10826 5/20 0.40
RARG P13631 5/20 0.40
MAPT P10636 4/20 0.36
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
CAPN1 P07384 2/20 0.36
PKM P14618 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
APP P05067 1/20 0.35
KDM4E B2RXH2 1/20 0.34
S1PR5 Q9H228 1/20 0.34
HPGD P15428 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7699617 1.00 GRIK1 (0.42) GRIK1GRIA1GRIA2GRIA3GRIA4
SCHEMBL18247318 0.87 GRIK1 (0.40) GRIK1GRIA1GRIA2GRIA3GRIA4
SCHEMBL7137570 0.85 RARB (0.53) RARARARBRARGMAPTNPC1
SCHEMBL20163299 0.85 RARB (0.53) RARARARBRARGMAPTNPC1
SCHEMBL7146567 0.85 RARB (0.53) RARARARBRARGMAPTNPC1
SCHEMBL7699620 0.79 RARA (0.39) RARARARBRARGNPC1RAB9A
SCHEMBL7140836 0.72 RARA (0.50) RARARARBRARGMAPTNPC1
SCHEMBL7140832 0.72 RARA (0.50) RARARARBRARGMAPTNPC1
SCHEMBL7143121 0.72 KMT2A (0.39) SMN1; SMN2LMNAKMT2A
SCHEMBL7139314 0.72 RARB (0.52) RARARARBRARGCYP3A4RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1212316-A2 BENZOPYRANS AND BENZOTHIOPYRANS AS RAR SELECTIVE RETINOID AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2002-06-12 EP disclosed
WO-2001014360-A2 BENZOPYRANS AND BENZOTHIOPYRANS AS RAR SELECTIVE RETINOID AGONISTS F. HOFFMAN-LA ROCHE AG (CH) 2001-03-01 WO disclosed