SCHEMBL7700759

SCHEMBL7700759

CC(COc1ccccc1Cl)N(C)CCc1ccc(N(OC(=O)/C=C/C(=O)O)S(C)(=O)=O)cc1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
CYP1A2 P05177 1/20 0.34
GAA P10253 1/20 0.34
CYP2C19 P33261 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HRH1 P35367 2/20 0.33
SIGMAR1 Q99720 2/20 0.33
LTB4R Q15722 2/20 0.33
LTB4R2 Q9NPC1 2/20 0.33
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL7700757 0.84 KCNH2 (0.44) CYP1A2CYP2C19
Fumaric Acid SCHEMBL7700761 0.84 KCNH2 (0.44) CYP1A2CYP2C19
SCHEMBL8286567 0.83 MEN1 (0.36) MEN1KMT2ACYP1A2CYP2C19KDM4E
SCHEMBL10589521 0.65 CNR2 (0.37) ALDH1A1
Hydrochloric Acid SCHEMBL7701317 0.65 KCNH2 (0.47) CYP1A2CYP2C19KDM4EALDH1A1SIGMAR1
Hydrochloric Acid SCHEMBL7702535 0.64 KCNH2 (0.47) CYP1A2CYP2C19KDM4EALDH1A1SIGMAR1
SCHEMBL7700726 0.63 CYP2D6 (0.44) CYP1A2GAACYP2C19ALDH1A1
Hydrochloric Acid SCHEMBL7700691 0.61 KCNH2 (0.48) CYP1A2CYP2C19KDM4EALDH1A1HPGD
SCHEMBL2008744 0.61 KCNH2 (0.47) CYP1A2CYP2C19KDM4EALDH1A1HPGD
Fumaric Acid SCHEMBL10921842 0.59 HRH1 (0.47) MEN1KMT2AKDM4EALDH1A1HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1037871-B1 NOVEL ANTIARRHYTHMIC COMPOUNDS GYOGYSZERKUTATO INTEZET (HU) 2002-07-03 EP disclosed
US-6265445-B1 CARDIOVASCULAR DISORDERS GYOGYSZERKUTATO INTEZET KFT (HU) 2001-07-24 US disclosed