SCHEMBL7700726

SCHEMBL7700726

CC(COc1ccccc1Cl)N(C)C(=O)Cc1ccc(NS(C)(=O)=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.44
OPRM1 P35372 1/20 0.44
OPRD1 P41143 1/20 0.44
OPRK1 P41145 1/20 0.44
ALDH1A1 P00352 1/20 0.42
KCNH2 Q12809 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP2C19 P33261 1/20 0.41
GAA P10253 1/20 0.41
ADRB2 P07550 1/20 0.40
ADRB1 P08588 1/20 0.40
ADRB3 P13945 1/20 0.40
EGFR P00533 2/20 0.40
ERBB2 P04626 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7696108 0.85 OPRK1 (0.42) CYP2D6OPRM1OPRD1OPRK1KCNH2
SCHEMBL7699534 0.81 KEAP1 (0.42) CYP2D6OPRM1OPRD1OPRK1ALDH1A1
SCHEMBL8213885 0.80 RORC (0.41) CYP2D6OPRM1OPRD1OPRK1ALDH1A1
Fumaric Acid SCHEMBL7700757 0.79 KCNH2 (0.44) CYP2D6KCNH2CYP1A2CYP3A4CYP2C9
Fumaric Acid SCHEMBL7700761 0.79 KCNH2 (0.44) CYP2D6KCNH2CYP1A2CYP3A4CYP2C9
SCHEMBL7886297 0.73 MEN1 (0.43) CYP1A2CYP2C19GAAADRB2ADRB1
SCHEMBL27446337 0.73 MEN1 (0.41) CYP1A2CYP2C19GAAADRB2ADRB1
SCHEMBL21895867 0.70 LMNA (0.41) ALDH1A1CYP1A2CYP2C19GAAEGFR
Hydrochloric Acid SCHEMBL7701317 0.69 KCNH2 (0.47) CYP2D6ALDH1A1KCNH2CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL7702535 0.68 KCNH2 (0.47) CYP2D6ALDH1A1KCNH2CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1140498-C Novel antiarrhythmic compounds ҩ���о�Ժ������ҵ 2004-03-03 CN disclosed
EP-1037871-B1 NOVEL ANTIARRHYTHMIC COMPOUNDS GYOGYSZERKUTATO INTEZET (HU) 2002-07-03 EP disclosed
US-6265445-B1 CARDIOVASCULAR DISORDERS GYOGYSZERKUTATO INTEZET KFT (HU) 2001-07-24 US disclosed
CN-1284941-A Novel antiarrhythmic compounds PHARMACEUTICAL RES INST PUBLIC (HU) 2001-02-21 CN disclosed