SCHEMBL8286567

SCHEMBL8286567

CC(CN(C)CCc1ccc(N(OC(=O)/C=C/C(=O)O)S(C)(=O)=O)cc1)Oc1ccccc1Cl

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
HPGD P15428 1/20 0.36
SLC6A9 P48067 1/20 0.34
NR1H4 Q96RI1 1/20 0.33
KCNH2 Q12809 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
MAPK1 P28482 1/20 0.33
CYP2C19 P33261 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HCAR2 Q8TDS4 1/20 0.32
LPAR1 Q92633 1/20 0.32
LPAR5 Q9H1C0 1/20 0.32
HRH1 P35367 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7700759 0.83 MEN1 (0.35) MEN1KMT2AHPGDCYP1A2CYP2C19
Fumaric Acid SCHEMBL7700757 0.67 KCNH2 (0.44) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
Fumaric Acid SCHEMBL7700761 0.67 KCNH2 (0.44) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL10589521 0.65 CNR2 (0.37) ALDH1A1HCAR2
Hydrochloric Acid SCHEMBL8216596 0.65 KCNH2 (0.50) HPGDKCNH2CYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL8205350 0.64 KCNH2 (0.49) HPGDKCNH2CYP1A2CYP3A4CYP2D6
SCHEMBL8213885 0.63 RORC (0.41) MEN1KMT2AHPGDKCNH2CYP1A2
Fumaric Acid SCHEMBL7316884 0.61 SLC6A9 (0.65) MEN1KMT2AHPGDSLC6A9CYP3A4
Maleic Acid SCHEMBL7316880 0.61 SLC6A9 (0.65) MEN1KMT2AHPGDSLC6A9CYP3A4
SCHEMBL6140360 0.61 KCNH2 (0.50) HPGDKCNH2CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1037871-A1 NOVEL ANTIARRHYTHMIC COMPOUNDS GYOGYSZERKUTATO INTEZET KFT. (HU) 2000-09-27 EP disclosed
WO-1999029655-A1 NOVEL ANTIARRHYTHMIC COMPOUNDS Gyógyszerkutató Intézet Kft. (HU) 1999-06-17 WO disclosed