SCHEMBL7702162

SCHEMBL7702162

CN(Cc1ccccc1)C(=O)Nc1ccc(-c2n[nH]c3c2Cc2ccccc2-3)cc1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDR P35968 6/20 0.55
CHEK1 O14757 8/20 0.53
CDK1 P06493 1/20 0.49
CDK2 P24941 1/20 0.49
MTOR P42345 2/20 0.47
KIT P10721 3/20 0.45
FLT1 P17948 3/20 0.45
TP53 P04637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7701942 0.87 CHEK1 (0.54) KDRCHEK1CDK1CDK2
SCHEMBL7700755 0.86 CHEK1 (0.52) KDRCHEK1CDK1CDK2
SCHEMBL7094008 0.84 CHEK1 (0.50) KDRCHEK1CDK1CDK2
SCHEMBL7095260 0.83 CHEK1 (0.58) KDRCHEK1CDK1CDK2
SCHEMBL7705309 0.82 KDR (0.69) KDRCHEK1CDK1CDK2
SCHEMBL7000769 0.81 CHEK1 (0.64) KDRCHEK1CDK1CDK2
SCHEMBL7698769 0.81 KDR (0.58) KDRCHEK1CDK1CDK2KIT
Hydrochloric Acid SCHEMBL7089690 0.80 CHEK1 (0.62) KDRCHEK1CDK1CDK2
SCHEMBL7697800 0.80 CHEK1 (0.57) KDRCHEK1CDK1CDK2
SCHEMBL7001943 0.80 CHEK1 (0.52) KDRCHEK1CDK1CDK2KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6462036-B1 INHIBITING SIGNAL TRANSDUCTION BY MODULATING ACTIVITY OF RECEPTOR AND NONRECEPTOR TYROSINE AND SERINE/THREONINE KINASES TO REGULATE AND MODULATE ABNORMAL OR INAPPROPRIATE CELL PROLIFERATION, DIFFERENTIATION, OR METABOLISM BASF AKTIENGESELLSCHAFT (DE) 2002-10-08 US disclosed