SCHEMBL7702655

SCHEMBL7702655

Nc1nccc2cc(CNC(=O)[C@@H]3CCCN3C(=O)[C@H](N)Cc3ccccc3)ccc12

nearest known ligand 0.65

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
F11 P03951 10/20 0.65
F2 P00734 7/20 0.65
F10 P00742 3/20 0.49
F12 P00748 3/20 0.49
PRSS1 P07477 3/20 0.49
PRSS2 P07478 3/20 0.49
F7 P08709 3/20 0.49
PRSS3 P35030 3/20 0.49
F9 P00740 1/20 0.49
KLKB1 P03952 2/20 0.49
KLK1 P06870 2/20 0.49
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
PKM P14618 1/20 0.48
CYP2C19 P33261 1/20 0.48
ALDH1A1 P00352 1/20 0.48
ROCK1 Q13464 1/20 0.47
OPRM1 P35372 1/20 0.46
OPRD1 P41143 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21429784 0.92 F11 (0.63) F11F2F10F12PRSS1
SCHEMBL24645591 0.92 F11 (0.63) F11F2F10F12PRSS1
Trifluoroacetic Acid SCHEMBL27886446 0.91 F11 (0.62) F11F2F10F12PRSS1
SCHEMBL3767038 0.88 F11 (0.65) F11F2F10F12PRSS1
SCHEMBL6438340 0.88 F11 (0.65) F11F2F10F12PRSS1
SCHEMBL7425868 0.88 F11 (0.58) F11F2F10F12PRSS1
SCHEMBL7147704 0.87 F11 (0.69) F11F2F10F12PRSS1
SCHEMBL29481406 0.87 F11 (0.56) F11F2F10F12PRSS1
SCHEMBL23013216 0.87 F11 (0.56) F11F2F10F12PRSS1
SCHEMBL23013213 0.87 F11 (0.56) F11F2F10F12PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6444672-B1 ORAL BIOVAILABILITY; INHIBITORS OF THROMBIN AND/OR FACTOR XA; SERINE PROTEASE INHIBITOR AKZO NOBEL N.V. (NL) 2002-09-03 US disclosed