SCHEMBL7702720

SCHEMBL7702720

CS(=O)(=O)Nc1ccc2[nH]cc(C3CCN(CCC4CCN(/C=C/C(=O)c5ccc(Cl)c(Cl)c5)CC4)CC3)c2c1

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 9/20 0.61
SLC2A1 P11166 1/20 0.48
HTR1D P28221 8/20 0.47
HTR1B P28222 6/20 0.45
DRD2 P14416 2/20 0.45
CHRM2 P08172 1/20 0.45
HTR6 P50406 2/20 0.45
HTR1A P08908 1/20 0.45
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45
HTR1E P28566 1/20 0.45
HTR1F P30939 1/20 0.45
HTR7 P34969 1/20 0.45
DRD3 P35462 1/20 0.45
HTR2B P41595 1/20 0.45
CCR5 P51681 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7696192 0.93 CCR2 (0.58) CCR2SLC2A1HTR1DHTR1BDRD2
SCHEMBL7702546 0.88 SLC2A1 (0.52) CCR2SLC2A1HTR1DHTR1BDRD2
SCHEMBL7694620 0.87 CCR2 (0.56) CCR2SLC2A1HTR1DHTR1BDRD2
SCHEMBL7700411 0.87 CCR2 (0.51) CCR2SLC2A1HTR1DHTR1BDRD2
SCHEMBL7699820 0.86 CCR2 (0.58) CCR2SLC2A1DRD2HTR6HTR1A
SCHEMBL7701607 0.84 SLC2A1 (0.58) CCR2SLC2A1HTR1DHTR1BDRD2
SCHEMBL7695961 0.83 HTR1D (0.54) CCR2HTR1DHTR1BDRD2CHRM2
SCHEMBL7700232 0.83 SLC2A1 (0.69) CCR2SLC2A1
SCHEMBL7700045 0.83 CCR2 (0.56) CCR2SLC2A1HTR1DHTR1BDRD2
SCHEMBL7699076 0.82 CCR2 (0.52) CCR2HTR1DHTR1BDRD2CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002079190-A1 3-SUBSTITUTED INDOLES AS CHEMOKINE ANTAGONISTS SMITHKLINE BEECHAM P.L.C. (GB) 2002-10-10 WO disclosed