SCHEMBL7702867

SCHEMBL7702867

O=C(Nc1ccc(-c2n[nH]c3c2Cc2ccccc2-3)cc1)c1ccc(F)cc1F

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 8/20 0.53
KDR P35968 2/20 0.52
CDK1 P06493 1/20 0.49
CDK2 P24941 1/20 0.49
ALDH1A1 P00352 2/20 0.45
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
KDM4E B2RXH2 1/20 0.45
MAPK1 P28482 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
AVPR2 P30518 1/20 0.44
GPR27 Q9NS67 1/20 0.44
SNCA P37840 1/20 0.43
MAPT P10636 1/20 0.43
PARP1 P09874 1/20 0.42
AURKA O14965 1/20 0.42
AURKB Q96GD4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7700585 0.92 CHEK1 (0.53) CHEK1KDRCDK1CDK2PARP1
SCHEMBL7697888 0.90 CHEK1 (0.57) CHEK1KDRCDK1CDK2ALDH1A1
SCHEMBL7095790 0.90 ALDH1A1 (0.49) CHEK1KDRALDH1A1AVPR2GPR27
SCHEMBL7696243 0.86 CHEK1 (0.57) CHEK1KDRCDK1CDK2ALDH1A1
SCHEMBL7702848 0.85 CHEK1 (0.54) CHEK1KDRCDK1CDK2NPC1
SCHEMBL7093397 0.85 CHEK1 (0.54) CHEK1KDRCDK1CDK2NPC1
SCHEMBL7091231 0.85 CHEK1 (0.56) CHEK1KDRCDK1CDK2AURKA
SCHEMBL7701201 0.82 CYP1A2 (0.49) CHEK1KDRNPC1RAB9AMAPT
SCHEMBL7094928 0.81 KDR (0.64) CHEK1KDRCDK1CDK2NPC1
SCHEMBL7701122 0.81 CHEK1 (0.48) CHEK1KDRCDK1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6462036-B1 INHIBITING SIGNAL TRANSDUCTION BY MODULATING ACTIVITY OF RECEPTOR AND NONRECEPTOR TYROSINE AND SERINE/THREONINE KINASES TO REGULATE AND MODULATE ABNORMAL OR INAPPROPRIATE CELL PROLIFERATION, DIFFERENTIATION, OR METABOLISM BASF AKTIENGESELLSCHAFT (DE) 2002-10-08 US disclosed