SCHEMBL7703480

SCHEMBL7703480

C/C=C/C(=O)C1CCC(c2ccccn2)CC1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 1/20 0.41
DRD4 P21917 11/20 0.40
DRD2 P14416 6/20 0.39
DRD3 P35462 3/20 0.39
HSD11B1 P28845 2/20 0.39
ADRA1D P25100 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36
KDM5A P29375 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7710548 1.00 HCRTR2 (0.41) HCRTR2DRD4DRD2DRD3HSD11B1
SCHEMBL7704805 0.82 HCRTR2 (0.38) HCRTR2
SCHEMBL7712965 0.82 KDM5A (0.37) KDM5A
SCHEMBL16803142 0.80 DRD4 (0.44) HCRTR2DRD4DRD2DRD3HSD11B1
SCHEMBL7710964 0.80 KDM4E (0.35) ADRA1A
SCHEMBL22999404 0.79 NPC1 (0.51) HCRTR2DRD4DRD2DRD3
Acetic Acid SCHEMBL29178492 0.78 ALDH1A1 (0.46) DRD4DRD2DRD3HSD11B1ADRA1D
SCHEMBL30131210 0.77 KMT2A (0.47) HCRTR2DRD4DRD2DRD3HSD11B1
SCHEMBL16803154 0.77 KMT2A (0.47) HCRTR2DRD4DRD2DRD3HSD11B1
Propionic Acid SCHEMBL29117403 0.77 DRD4 (0.46) HCRTR2DRD4DRD2DRD3ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011131596-A1 HETEROARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES AS VASOPRESSIN V1A RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2011-10-27 WO disclosed