SCHEMBL7712965

SCHEMBL7712965

C/C=C/C(=O)C1CCC(c2cccnn2)CC1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 1/20 0.37
CCR2 P41597 1/20 0.32
HDAC4 P56524 1/20 0.31
PDE4A P27815 2/20 0.30
PDE4B Q07343 2/20 0.30
PDE4C Q08493 2/20 0.30
PDE4D Q08499 2/20 0.30
TYK2 P29597 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7710548 0.82 HCRTR2 (0.41) KDM5A
SCHEMBL7703480 0.82 HCRTR2 (0.41) KDM5A
SCHEMBL2563182 0.79 NPC1 (0.46) KDM5AHDAC4PDE4APDE4BPDE4C
SCHEMBL2563184 0.79 NPC1 (0.46) KDM5AHDAC4PDE4APDE4BPDE4C
SCHEMBL29765569 0.76
SCHEMBL16060787 0.76
SCHEMBL7707988 0.75 CYP11B2 (0.50)
SCHEMBL7704805 0.75 HCRTR2 (0.38) HDAC4
SCHEMBL2563797 0.74 P2RX7 (0.44) KDM5AHDAC4
SCHEMBL2560138 0.74 GAA (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011131596-A1 HETEROARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES AS VASOPRESSIN V1A RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2011-10-27 WO disclosed