SCHEMBL7703616

SCHEMBL7703616

COc1ccc(I)c2c1oc1cncnc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
MAPT P10636 4/20 0.34
P2RX3 P56373 1/20 0.34
P2RX2 Q9UBL9 1/20 0.34
MGAM O43451 1/20 0.33
TSHR P16473 3/20 0.33
HSD17B10 Q99714 3/20 0.33
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33
CLK1 P49759 1/20 0.32
IRAK4 Q9NWZ3 2/20 0.31
CYP19A1 P11511 2/20 0.31
CYP17A1 P05093 1/20 0.31
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
IDO1 P14902 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL73148 0.83 MAPT (0.38) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL73387 0.80 KDM4E (0.36) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL75224 0.79 PDE4A (0.43) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL72743 0.74 MAOA (0.49) MAPTTSHRHSD17B10ALDH1A1KDM4E
SCHEMBL2560611 0.71 PDE4A (0.42) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL20457804 0.71 SMN1; SMN2 (0.30) SMN1; SMN2
SCHEMBL74891 0.71 PDE4D (0.63) PDE4APDE4BPDE4CPDE4D
SCHEMBL7650714 0.65 NPC1 (0.42) HSD17B10ALDH1A1CYP19A1LMNACYP1A2
SCHEMBL26771405 0.64 SMN1; SMN2 (0.42) MAPTTSHRHSD17B10ALDH1A1KDM4E
SCHEMBL25662814 0.63 CCR1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011132051-A2 TRICYCLE COMPOUNDS AS PHOSPHODIESTERASE-10 INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2011-10-27 WO disclosed