SCHEMBL7704152

SCHEMBL7704152

CCC(Cc1ccccc1)=C(c1ccccc1)c1ccc(OCCN(C)C)cc1.CCC(Cc1ccccc1)=C(c1ccccc1)c1ccc(OCCN(CC)CC)cc1.CCC(Cc1ccccc1)=C(c1ccccc1)c1ccc(OCCN2CCCC2)cc1.CCC(Cc1ccccc1)=C(c1ccccc1)c1ccc(OCCN2CCCCC2)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 7/20 0.70
PSMB1 P20618 9/20 0.60
PSMB5 P28074 8/20 0.60
PSMB2 P49721 4/20 0.60
ESR2 Q92731 3/20 0.54
PDE1A P54750 2/20 0.54
PDE1B Q01064 2/20 0.54
PDE1C Q14123 2/20 0.54
MAPT P10636 2/20 0.52
MEN1 O00255 1/20 0.52
NPC1 O15118 1/20 0.52
NR1I2 O75469 1/20 0.52
PRKD3 O94806 1/20 0.52
ABCB11 O95342 1/20 0.52
EGFR P00533 1/20 0.52
GBA1 P04062 1/20 0.52
NR3C1 P04150 1/20 0.52
ERBB2 P04626 1/20 0.52
TP53 P04637 1/20 0.52
PRKCG P05129 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7603635 0.89 ESR1 (0.88) ESR1PSMB1PSMB5PSMB2ESR2
SCHEMBL7597039 0.88 ESR1 (0.89) ESR1PSMB1PSMB5PSMB2ESR2
SCHEMBL7602293 0.84 ESR1 (0.65) ESR1PSMB1PSMB5ESR2MAPT
SCHEMBL7597053 0.83 ESR1 (0.68) ESR1PSMB1PSMB5ESR2PDE1A
SCHEMBL7598246 0.83 ESR1 (1.00) ESR1PSMB1PSMB5PSMB2ESR2
SCHEMBL7598249 0.83 ESR1 (1.00) ESR1PSMB1PSMB5PSMB2ESR2
SCHEMBL23266951 0.80 PSMB1 (0.87) ESR1PSMB1PSMB5PSMB2ESR2
SCHEMBL7601189 0.79 ESR1 (0.74) ESR1PSMB1PSMB5PSMB2ESR2
SCHEMBL7602726 0.78 ESR1 (0.72) ESR1PSMB1PSMB5ESR2MAPT
SCHEMBL7602724 0.78 ESR1 (0.72) ESR1PSMB1PSMB5ESR2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002066415-A2 NON-STEROIDAL MODULATORS OF ESTROGEN RECEPTORS THE PROVOST, FELLOWS AND SCHOLARS OF THE COLLEGE OF THE HOLY AND UNDIVIDED TRINITY OF QUEEN ELIZABETH NEAR DUBLIN (IE) 2002-08-29 WO claimed