SCHEMBL7704154

SCHEMBL7704154

CN(C)CCCOc1ncc(C(=O)O)c(-c2ccc(F)cc2Cl)n1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
PAICS P22234 2/20 0.37
RXRA P19793 1/20 0.37
RXRB P28702 1/20 0.37
CDC7 O00311 1/20 0.36
DBF4 Q9UBU7 1/20 0.36
ALDH1A1 P00352 3/20 0.36
LMNA P02545 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
EIF4E P06730 1/20 0.36
PRKAG1 P54619 1/20 0.35
PRKAA1 Q13131 1/20 0.35
PRKAB1 Q9Y478 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CCNT1 O60563 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6016492 0.95 PAICS (0.41) KDM4ESMN1; SMN2PAICSRXRARXRB
SCHEMBL6016618 0.92 MEN1 (0.35) KDM4ESMN1; SMN2PAICSRXRARXRB
Dimethylaminoethanol SCHEMBL6016393 0.91 PAICS (0.39) KDM4ESMN1; SMN2PAICSRXRARXRB
SCHEMBL6016402 0.85 MAPK14 (0.43) KDM4ESMN1; SMN2ALDH1A1KMT2A
SCHEMBL6016397 0.85 CDC7 (0.39) KDM4EPAICSCDC7DBF4ALDH1A1
SCHEMBL6016620 0.84 ACHE (0.36) KDM4ESMN1; SMN2PAICSCDC7DBF4
SCHEMBL6016572 0.80 MAPK14 (0.48) KDM4ESMN1; SMN2PAICSALDH1A1KMT2A
SCHEMBL6016703 0.78 MAPK14 (0.39) KDM4EALDH1A1MEN1KMT2A
SCHEMBL6016414 0.78 PRKAB2 (0.47) KDM4EALDH1A1PRKAG1PRKAA1PRKAB1
SCHEMBL6016503 0.78 KDM4E (0.41) KDM4ESMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1166643-C 4-phenyl-pyrimidine derivatives - 2004-09-15 CN disclosed
CN-1353697-A 4-phenyl-pyrimidine derivatives HOFFMANN LA ROCHE (CH) 2002-06-12 CN disclosed
EP-1187815-A1 4-PHENYL-PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-03-20 EP disclosed
US-6274588-B1 NEUROKININ OR SUBSTANCE P ANTAGONISTS; CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDES; ANTIDEPRESSANTS, ANXIOLYTIC AGENTS HOFFMANN-LA ROCHE INC. 2001-08-14 US disclosed
WO-2000073279-A1 4-PHENYL-PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-12-07 WO disclosed