SCHEMBL7705200

SCHEMBL7705200

COc1ccc(-c2c(C(F)(F)F)c[c]cc2C(F)(F)F)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 2/20 0.50
AR P10275 2/20 0.50
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
KDM4E B2RXH2 2/20 0.43
GLA P06280 1/20 0.43
MAPT P10636 1/20 0.43
CYP1A2 P05177 1/20 0.42
ACHE P22303 1/20 0.41
ENPP1 P22413 1/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
NT5E P21589 1/20 0.39
PTGS2 P35354 2/20 0.39
ESR2 Q92731 1/20 0.38
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7702032 0.79 AR (0.46) ARCYP11B1CYP11B2KDM4EGLA
SCHEMBL7955020 0.78 PGR (0.47) PGRARCYP11B1CYP11B2KDM4E
SCHEMBL7704882 0.77 KDM4E (0.37) ARKDM4EMAPTACHEENPP1
SCHEMBL7701995 0.76 CYP11B1 (0.37) CYP11B1CYP11B2KDM4EMAPT
SCHEMBL7465724 0.75 KIF11 (0.41) CYP11B2KDM4EGLAMAPTACHE
SCHEMBL730765 0.73 CA12 (0.46) KDM4EMAPTACHECA12CA1
SCHEMBL20323072 0.71 CA1 (0.69) KDM4EMAPTACHECA12CA1
SCHEMBL2290039 0.70 AR (0.33) PGRAR
SCHEMBL5803017 0.69 ABL1 (0.55) PGRARMAPTENPP1MEN1
SCHEMBL7705198 0.69 PGR (0.44) PGRARCYP11B1CYP11B2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242399-A1 $g(a)-ARYLETHYLPIPERAZINE DERIVATIVES AS NEUROKININ ANTAGONISTS UCB S.A. (BE) 2002-09-25 EP disclosed
WO-2001046167-A1 α-ARYLETHYLPIPERAZINE DERIVATIVES AS NEUROKININ ANTAGONISTS UCB, S.A. (BE) 2001-06-28 WO disclosed