SCHEMBL7705631

SCHEMBL7705631

CCC1CCCCN1CCn1c(C2CCCN2)nc2c(C(N)=O)cccc21

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 19/20 0.47
PARP2 Q9UGN5 7/20 0.42
PARP3 Q9Y6F1 1/20 0.42
TAAR1 Q96RJ0 1/20 0.37
MAP4K4 O95819 1/20 0.37
CSF1R P07333 1/20 0.37
PIM1 P11309 1/20 0.37
CLK2 P49760 1/20 0.37
MAP4K2 Q12851 1/20 0.37
DYRK1A Q13627 1/20 0.37
MINK1 Q8N4C8 1/20 0.37
AURKB Q96GD4 1/20 0.37
MAP4K5 Q9Y4K4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5620585 0.98 PARP1 (0.47) PARP1PARP2PARP3MAP4K4CSF1R
SCHEMBL7700402 0.91 PARP1 (0.49) PARP1PARP2PARP3
SCHEMBL7041448 0.88 TAAR1 (0.36) PARP1TAAR1
SCHEMBL5621352 0.87 PARP1 (0.52) PARP1PARP2
SCHEMBL5621642 0.86 PARP1 (0.48) PARP1PARP2PARP3MAP4K4CSF1R
SCHEMBL7706378 0.85 PARP1 (0.49) PARP1PARP2PARP3DYRK1A
SCHEMBL5619993 0.85 PARP1 (0.53) PARP1PARP2PARP3PIM1AURKB
SCHEMBL5621834 0.85 PARP1 (0.52) PARP1PARP2PARP3
SCHEMBL5620530 0.84 PARP1 (0.57) PARP1PARP2
SCHEMBL7705473 0.83 PARP1 (0.56) PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6448271-B1 SUCH AS 2-(PIPERIDIN-4-YL)BENZIMIDAZOLE-4-CARBOXAMIDE; INHIBITORS OF ENZYME POLY(ADP-RIBOSE)POLYMERASE; IMPROVED WATER SOLUBILITY BASF AKTIENGESELLSCHAFT (DE) 2002-09-10 US disclosed