SCHEMBL7705812

SCHEMBL7705812

FC(F)(F)c1cc(-c2cccc3ccccc23)cc(C(F)(F)F)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.43
CYP1A1 P04798 1/20 0.43
CYP1B1 Q16678 1/20 0.43
CNR2 P34972 2/20 0.41
P2RX1 P51575 1/20 0.41
P2RX3 P56373 1/20 0.41
P2RX4 Q99571 1/20 0.41
P2RX7 Q99572 1/20 0.41
FNTA P49354 1/20 0.41
FNTB P49356 1/20 0.41
MCL1 Q07820 1/20 0.41
ACMSD Q8TDX5 1/20 0.41
HTR1A P08908 1/20 0.40
HTR7 P34969 1/20 0.40
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA9 Q16790 2/20 0.40
CNR1 P21554 1/20 0.40
HDAC8 Q9BY41 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31230608 0.87 CYP1A1 (0.40) CYP1A2CYP1A1CYP1B1CNR2P2RX1
SCHEMBL22993088 0.86 CNR1 (0.42) CYP1A2CYP1A1CYP1B1CNR2P2RX1
SCHEMBL26547948 0.86 CA12 (0.46) CYP1A2CYP1A1CYP1B1P2RX1P2RX3
SCHEMBL26548388 0.86 CA12 (0.46) CYP1A2CYP1A1CYP1B1P2RX1P2RX3
SCHEMBL26548881 0.85 CA12 (0.45) CYP1A2CYP1A1CYP1B1P2RX1P2RX3
SCHEMBL26548570 0.85 CA12 (0.45) CYP1A2CYP1A1CYP1B1P2RX1P2RX3
SCHEMBL13268400 0.85 CNR1 (0.39) CYP1A2CYP1A1CYP1B1CNR2P2RX1
SCHEMBL28224945 0.83 KIF11 (0.52) CNR2CA12CA1CA2CA9
SCHEMBL29805137 0.81 CYP11B1 (0.40) CYP1A2CYP1A1CYP1B1CNR2P2RX1
SCHEMBL31139510 0.80 CES1 (0.50) CYP1A2CYP1A1CYP1B1CNR2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242399-A1 $g(a)-ARYLETHYLPIPERAZINE DERIVATIVES AS NEUROKININ ANTAGONISTS UCB S.A. (BE) 2002-09-25 EP disclosed
WO-2001046167-A1 α-ARYLETHYLPIPERAZINE DERIVATIVES AS NEUROKININ ANTAGONISTS UCB, S.A. (BE) 2001-06-28 WO disclosed