SCHEMBL7705836

SCHEMBL7705836

Nc1nccnc1C1CNC1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 3/20 0.42
CHRNA3 P32297 3/20 0.42
CHRNB2 P17787 3/20 0.42
CHRNA4 P43681 3/20 0.42
CHRNA1 P02708 1/20 0.42
ESR1 P03372 1/20 0.42
CHRNG P07510 1/20 0.42
CHRNB1 P11230 1/20 0.42
CHRNA5 P30532 1/20 0.42
CHRNA7 P36544 1/20 0.42
HTR3A P46098 1/20 0.42
CHRND Q07001 1/20 0.42
CHRNA2 Q15822 1/20 0.42
HRH3 Q9Y5N1 1/20 0.37
TNK2 Q07912 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9900635 0.84 HTR3A (0.38) CHRNB4CHRNA3CHRNB2CHRNA4CHRNA1
SCHEMBL9901829 0.84 HTR3A (0.38) CHRNB4CHRNA3CHRNB2CHRNA4CHRNA1
SCHEMBL30673624 0.84 HTR3A (0.38) CHRNB4CHRNA3CHRNB2CHRNA4CHRNA1
SCHEMBL9900173 0.81 BTK (0.46)
SCHEMBL9900029 0.81 BTK (0.46)
SCHEMBL9900636 0.79 NEK2 (0.34)
SCHEMBL30154873 0.79 NEK2 (0.34)
SCHEMBL28076460 0.79 HRH4 (0.41) HRH3TNK2
SCHEMBL14440475 0.75 CHRNB2 (0.57) CHRNB4CHRNA3CHRNB2CHRNA4CHRNA1
SCHEMBL7699577 0.74 CHRNB2 (0.42) CHRNB4CHRNA3CHRNB2CHRNA4CHRNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011143365-A1 NITROGEN HETEROCYCLIC COMPOUNDS USEFUL AS PDE10 INHIBITORS AMGEN INC. (US) 2011-11-17 WO disclosed