SCHEMBL7706770

SCHEMBL7706770

CC(=O)Nc1ccc2c3c(cccc13)C(=O)OC2=O

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.63
ALDH1A1 P00352 4/20 0.63
GAA P10253 3/20 0.63
TYMS P04818 4/20 0.54
HPGD P15428 2/20 0.54
MAPT P10636 1/20 0.54
RXFP1 Q9HBX9 1/20 0.47
MAOA P21397 1/20 0.45
KMT2A Q03164 4/20 0.44
MEN1 O00255 3/20 0.44
USP2 O75604 2/20 0.44
KEAP1 Q14145 1/20 0.44
NFE2L2 Q16236 1/20 0.44
HSD17B10 Q99714 1/20 0.44
BLM P54132 1/20 0.44
PARP14 Q460N5 2/20 0.43
CASP3 P42574 1/20 0.42
GPR35 Q9HC97 1/20 0.42
GLA P06280 1/20 0.42
PABPC1 P11940 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8062355 0.83 KDM4E (0.61) KDM4EALDH1A1GAAHPGDMAPT
SCHEMBL5964469 0.82 ALDH1A1 (0.71) KDM4EALDH1A1GAAHPGDMAPT
SCHEMBL7709637 0.81 TYMS (0.48) KDM4EALDH1A1GAATYMSHPGD
SCHEMBL9077602 0.81 TYMS (0.44) KDM4EALDH1A1GAATYMSHPGD
SCHEMBL9437196 0.79 ALDH1A1 (0.67) KDM4EALDH1A1GAAMAPTKMT2A
SCHEMBL28655617 0.77 KDM4E (1.00) KDM4EALDH1A1GAAHPGDMAPT
SCHEMBL2134658 0.77 TYMS (0.56) KDM4EALDH1A1GAATYMSMAPT
SCHEMBL9437176 0.76 ALDH1A1 (0.64) KDM4EALDH1A1GAAMAPTKMT2A
SCHEMBL11809469 0.76 TYMS (0.51) KDM4EALDH1A1GAATYMSHPGD
SCHEMBL7706686 0.76 TYMS (0.44) KDM4EALDH1A1GAATYMSKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362181-B1 BACTERICIDES; ENZYME INHIBITORS; ANTITUMOR AGENTS WARNER-LAMBERT COMPANY 2002-03-26 US disclosed
US-6177423-B1 N-(HYDROXY OR PROTECTED HYDROXY)-BENZO(DE)ISOQUINOLINE-1,3-DIONE DERIVATIVES; BACTERIAL DNA GYRASE AND DNA TOPOISOMERASE INHIBITORS USEFUL FOR ANTIBACTERIAL AGENTS HAVING REDUCED DRUG RESISTANCE AND REDUCED SIDE EFFECTS WARNER-LAMBERT COMPANY 2001-01-23 US disclosed
EP-0939754-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1999-09-08 EP disclosed
WO-1998019648-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1998-05-14 WO disclosed
US-4210757-A Novel naphthoylene-perinones disperse dyestuffs CIBA-GEIGY CORPORATION (US) 1980-07-01 US disclosed
US-4067889-A 2-CYANO-3-AMINO-BENZANTHRONES AS PRECURSORS CIBA-GEIGY CORPORATION (US) 1978-01-10 US disclosed
US-3970675-A ANTHRONE-AMIDINE CIBA-GEIGY CORPORATION (US) 1976-07-20 US disclosed