SCHEMBL7709637

SCHEMBL7709637

CC(=O)Nc1cc2c3c(cccc3c1Cl)C(=O)OC2=O

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TYMS P04818 3/20 0.48
KDM4E B2RXH2 5/20 0.44
ALDH1A1 P00352 4/20 0.44
GAA P10253 3/20 0.44
MAOA P21397 1/20 0.43
PARP14 Q460N5 4/20 0.43
CASP3 P42574 1/20 0.41
GPR35 Q9HC97 1/20 0.40
GLA P06280 1/20 0.40
HPGD P15428 2/20 0.40
HSD17B10 Q99714 2/20 0.40
HSP90AA1 P07900 2/20 0.39
HSP90AB1 P08238 2/20 0.39
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9077602 0.84 TYMS (0.44) TYMSKDM4EALDH1A1GAAMAOA
SCHEMBL7706770 0.81 KDM4E (0.63) TYMSKDM4EALDH1A1GAAMAOA
SCHEMBL7706744 0.76 ALDH1A1 (0.46) KDM4EALDH1A1GAAMAOAPARP14
SCHEMBL7706686 0.76 TYMS (0.44) TYMSKDM4EALDH1A1GAAHSP90AA1
SCHEMBL7709794 0.75 TYMS (0.66) TYMSKDM4EALDH1A1HPGDMAPT
SCHEMBL7706710 0.74 TYMS (0.45) TYMSKDM4EALDH1A1GAAMAOA
SCHEMBL7709571 0.72 TYMS (0.57) TYMSKDM4EALDH1A1HPGDMAPT
SCHEMBL7703727 0.72 TYMS (0.45) TYMSKDM4EGAAHPGDMAPT
SCHEMBL11412153 0.71 ALDH1A1 (0.47) KDM4EALDH1A1GAAMAOAPARP14
SCHEMBL9079791 0.70 KLK7 (0.71) TYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362181-B1 BACTERICIDES; ENZYME INHIBITORS; ANTITUMOR AGENTS WARNER-LAMBERT COMPANY 2002-03-26 US disclosed
US-6177423-B1 N-(HYDROXY OR PROTECTED HYDROXY)-BENZO(DE)ISOQUINOLINE-1,3-DIONE DERIVATIVES; BACTERIAL DNA GYRASE AND DNA TOPOISOMERASE INHIBITORS USEFUL FOR ANTIBACTERIAL AGENTS HAVING REDUCED DRUG RESISTANCE AND REDUCED SIDE EFFECTS WARNER-LAMBERT COMPANY 2001-01-23 US disclosed
EP-0939754-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1999-09-08 EP disclosed
WO-1998019648-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1998-05-14 WO disclosed